Research Group Publications

 
  • Yeware Amar, Agrawal Sonia And Sarkar Dhiman., A high content screening assay for identifying inhibitors against active and dormant state intracellular Mycobacterium tuberculosis, Journal of Microbiological Methods., 164, 105687 (2019).
  • Yeware Amar , Gample Suwarna, Agrawal Sonia And Sarkar Dhiman, Using diphenyleneiodonium to induce a viable but non-culturable phenotype in Mycobacterium tuberculosis and its metabolomics analysis, PLoS One., 14:8, e0220628 (2019).
  • Gample Suwarna, Agrawal Sonia And Sarkar Dhiman, Evidence of nitrite acting as a stable and robust inducer of non-cultivability in Mycobacterium tuberculosis with physiological relevance, Scientific reports., 9:1, 9261 (2019).
  • Uttam B Karale, Vagolu Siva Krishna, E Vamshi Krishna, Amit S Choudhari, Manjulika Shukla, Vikas R Gaikwad, B Mahizhaveni, Sidharth Chopra, Sunil Misra, Dhiman Sarkar, Dharmarajan Sriram, VN Azger Dusthackeer And Haridas B Rode, Synthesis and biological evaluation of 2, 4, 5-trisubstituted thiazoles as antituberculosis agents effective against drug-resistant tuberculosis, European journal of medicinal chemistry., , (2019).
  • Vikas Shinde, Pramod Mahulikar, Pravin C Mhaske, Shakti Chakraborty, Amit Choudhari, Siddharth Phalle, Prafulla Choudhari And Dhiman Sarkar, Synthesis and antimycobacterial evaluation of new 5-(1-benzyl-1H-1,2,3-triazol-4-yl)-4-methyl-2-arylthiazole derivatives, Medicinal Chemistry Research., 28, 805 - 819 (2019).
  • Sushma J Takate, Abhijit D Shinde, Bhausaheb K Karale, Hemant Akolkar, Laxman Nawale, Dhiman Sarkar And Pravin C Mhaske, Thiazolyl-pyrazole derivatives as potential antimycobacterial agents, Bioorganic & medicinal chemistry letters., 29, 1199 - 1202 (2019).
  • Atmaram Upare A, Gadekar PK, Sivaramakrishnan H, Naik N3, Khedkar VM, Sarkar D, Choudhari A And Mohana Roopan S., Design and Synthesis of 2?Amino?thiophene?proline?conjugates and Their Anti?tubercular Activity against Mycobacterium Tuberculosis H37Ra, Bioorg Chem., 86, 507 - 512 (2019), DOI:doi: 10.1016/j.bioorg.2019.01.054.
  • Amarsinh R Deshmukh, Sambhaji T Dhumal, Laxman U Nawale, Vijay M Khedkar, Dhiman Sarkar And Ramrao A Mane, Dicationic liquid mediated synthesis of tetrazoloquinolinyl methoxy phenyl 4-thiazolidinones and their antibacterial and antitubercular evaluation, Synthetic Communications., , 1 - 15 (2019).
  • Yeware Amar And Sarkar Dhiman , Novel red fluorescence protein based microplate assay for drug screening against dormant Mycobacterium tuberculosis by using paraffin, Tuberculosis., 110, 15 - 19 (2018), DOI:https://doi.org/10.1016/j.tube.2018.02.008.
  • Macchindra S Tambe, Amit Choudhari, Dhiman Sarkar, Jaiprakash Sangshetti, Rajesh Patil And Somnath S Gholap, Design, Synthesis and Biological Screening of Novel 1, 3, 4?Oxadiazoles as Antitubercular Agents, ChemistrySelect., 3;47, 13304 - 13310 (2018).
  • TS Chitre, SM Patil, AG Sujalegaonkar, KD Asgaonkar, VM Khedkar, DR Garud, PC Jha, SY Gaikwad, SS Kulkarni, A Choudhari And D Sarkar, Non nucleoside reverse transcriptase inhibitors, molecular docking studies and antitubercular activity of thiazolidin-4-one derivatives, Current computer-aided drug design., , (2018).
  • Hemlata M Mali, Sandip S Sabale, Mariam S Degani, Rachana Borkute, Amit S Choudhari, Dhiman Sarkar, Vagolu Siva Krishna And Dharmarajan Sriram, Rational design of coumarin derivatives as antituberculosis agents, Future medicinal chemistry., 10;20, 2431 - 2444 (2018).
  • Ashruba B Danne, Amit S Choudhari, Dhiman Sarkar, Jaiprakash N Sangshetti, Vijay M Khedkar And Bapurao B Shingate, Synthesis and biological evaluation of novel triazole-biscoumarin conjugates as potential antitubercular and anti-oxidant agents, Research on Chemical Intermediates., 44;10, 6283 - 6310 (2018).
  • Nishant K Rasal, Rahul B Sonawane, Amit S Choudhari, Shakti S Chakraborty, Dhiman D Sarkar And Sangeeta V Jagtap, Novel 2,4?Dimethyl?5?((E)?3?phenyl?3?oxoprop?1?enyl)?1H?pyrrole?3?carboxylic Acid Derivatives: New Leads in Cancer and Bacterial Chemotherapy, ChemistrySelect., 3;33, 9571 - 9575 (2018).
  • Rakhi Gawali, Jay Trivedi, Sujit Bhansali, Raghunath Bhosale, Dhiman Sarkar And Debashis Mitra, Design, synthesis, docking studies and biological screening of 2-thiazolyl substituted-2, 3-dihydro-1H-naphtho [1, 2-e][1, 3] oxazines as potent HIV-1 reverse transcriptase …, European journal of medicinal chemistry., 157, 310 - 319 (2018).
  • Urja Nimbalkar, Julio Seijas, Rachna Borkute, Manoj Damale, Jaiprakash Sangshetti, Dhiman Sarkar And Anna Nikalje, Ultrasound Assisted Synthesis of 4-(Benzyloxy)-N-(3-chloro-2-(substitutedphenyl)-4-oxoazetidin-1-yl) Benzamide as Challenging Anti-Tubercular Scaffold, Molecules., 23;8, 1945 (2018).
  • Yogesh Patil, Ramesh Shingare, Amit Choudhari, Rachana Borkute, Dhiman Sarkar And Balaji R Madje, Synthesis and biological evaluation of some new tricyclic pyrrolo[3,2?e]tetrazolo[1,5?c]pyrimidine derivatives as potential antitubercular agents, Archiv der Pharmazie., 351;8, 18000040 (2018).
  • MH Shaikh, DD Subhedar, L Nawale, D Sarkar, FAK Khan, J Sangshetti And BB Shingate, Novel Benzylidenehydrazide-1, 2, 3-Triazole conjugates as Antitubercular Agents: Synthesis and Molecular Docking, Mini reviews in medicinal chemistry., , (2018).
  • Hitendra Joshi, Dhiman Sarkar, Nirav Shah And Nisheeth C. Desai and Krunalsinh ..., One Pot Synthesis and Biological Evaluation of Some New Pyridine-3,5-dicarbonitrile Derivatives, Chemistrselect., 3, 3374 (2018).
  • Govind S Bhosle, Laxman Nawale, Amar M Yeware, Dhiman Sarkar And Moneesha Fernandes, Antibacterial and anti-TB tat-peptidomimetics with improved efficacy and half-life, European journal of medicinal chemistry., 152, 358 - 369 (2018).
  • Vikas Shinde, Pramod Mahulikar, Pravin Mhaske, Laxman Nawale And Dhiman Sarkar, Synthesis and biological evaluation of new 2-aryl-4-((4-aryl-1H-1,2,3-triazol-1-yl)methyl)thiazole derivatives, Research on Chemical Intermediates., 44, 1247 - 1260 (2018), DOI:https://doi.org/10.1007/s11164-017-3164-4.
  • Mahendra A. Wagh, Dr. Sachin B. Baravkar, Dr. Ganesh S. Jedhe, Rachana Borkute, Dr. Amit S. Choudhari, Dr. Dhiman Sarkar And Dr. Gangadhar J. Sanjayan, Design and Synthesis of 2-Amino-thiophene-Tethered Ureidopenicillin Analogs with Potent Antibacterial and Antitubercular activity, Chemistry Select., 3, 3122 - 3126 (2018), DOI:https://doi.org/10.1002/slct.201800027.
  • N. C. Desai, Amit Trivedi, Hardik Somani, Krunalsinh A. Jadeja, Darshita Vaja, Laxman Nawale, Vijay Khedkar And Dhiman Sarkar, Synthesis, biological evaluation, and molecular docking studies of pyridine clubbed 1,3,4-oxadiazoles as potential antituberculars, Synthetic Communications An International Journal for Rapid Communication of Synthetic Organic Chemistry., 48, 524 - 540 (2018), DOI:https://doi.org/10.1080/00397911.2017.1410892.
  • Somnath Gholap, Macchindra Tambe, Laxman Nawale, Dhiman Sarkar, Jaiprakash Sangshetti And Manoj Damale, Design, synthesis, and pharmacological evaluation of fluorinated azoles as anti-tubercular agents, ArchPharm., 351, (2018), DOI:https://doi.org/10.1002/ardp.201700294.
  • Ninad V. Puranik, Pratibha Srivastava, Sagar Swami, Amit Choudhari And Dhiman Sarkar, Molecular modeling studies and in vitro screening of dihydrorugosaflavonoid and its derivatives against Mycobacterium tuberculosis, RSC Advances., 8, 10634 - 10643 (2018), DOI:10.1039/C8RA00636A.
  • Amol S. Kotmale, Ekta Sangtani, Rajesh G. Gonnade, Dhiman Sarkar, Sachin Burade, Pattuparambil R. Rajamohanan And Gangadhar J. Sanjayan, Conformational studies of Ant-Pro motif-incorporated cyclic peptides: gramicidine S and avellanin, New Journal of Chemistry., 42, 1197 - 1201 (2018), DOI:10.1039/C7NJ03701E.
  • Yogesh Patil, Ramesh Shingare, Shakti Chakraborty, Rachana Borkute, Dhiman Sarkar And Balaji Madje, Synthesis and biological evaluation of some bicyclic [2-(2,4-dimethylphenylthio)phenyl] aniline and its amide derivatives as potential antitubercular agents, Journal of Chemical Sciences., 130, (2018), DOI:https://doi.org/10.1007/s12039-018-1424-5.
  • Bapurao B. Shingate, Ashruba Danne, Amit Choudhari, Shakti Chakraborty, Dhiman Sarkar And Vijay Khedkar, Triazole-Diindolylmethane Conjugates as New Antitubercular Agents: Synthesis, Bioevaluation and Molecular Docking, Med. Chem. Comm., , (2018), DOI:10.1039/C8MD00055G.
  • Mahesh M. Pisal, Ritesh A. Annadate, Meghana C. Athalye, Dipak Kumar, Subhash P. Chavan, Dhiman Sarkar And Hanumant B. Borate, Synthesis and cell imaging applications of fluorescent mono/di/tri-heterocyclyl-2,6-dicyanoanilines, Bioorganic & Medicinal Chemistry Letters., , (2017), DOI:10.1016/j.bmcl.2016.12.074.
  • Neha Tiwari, Laxman Nawale, Dhiman Sarkar And Manohar V. Badiger, Carboxymethyl Cellulose-Grafted Mesoporous Silica Hybrid Nanogels for Enhanced Cellular Uptake and Release of Curcumin, Gels., 3, 8 (2017), DOI:https://doi.org/10.3390/gels3010008.
  • Yogita K. Abhale, Abhijit D. Shinde, Keshav K. Deshmukh, Laxman Nawale, Dhiman Sarkar, Prafulla B. Choudhari, Santosh S. Kumbhar And Pravin C. Mhaske, Synthesis, antimycobacterial screening and molecular docking studies of 4-aryl-4'-methyl-2'-aryl-2,5-bisthiazole derivates, Medicinal Chemistry Research., 26, 2889 - 2899 (2017), DOI:https://doi.org/10.1007/s00044-017-1988-5.
  • Yogita K. Abhale, Abhijit Shinde, Keshav K. Deshmukh, Laxman Nawale, Dhiman Sarkar And Pravin Mhaske, Synthesis, antitubercular and antimicrobial potential of some new thiazole substituted thiosemicarbazide derivatives, Medicinal Chemistry Research., 26, 2557 - 2567 (2017), DOI:https://doi.org/10.1007/s00044-017-1955-1.
  • Sambhaji T. Dhumal, Amarsinh R. Deshmukh, Lalit D. Khillare, Manisha Arkile, Dhiman Sarkar And Ramrao A. Mane, Synthesis and Antitubercular activity of New Thiazolidinones with Pyrazinyl and Thiazolyl Scaffolds, Journal of Heterocyclic Chemistry., 54, 125 - 130 (2017), DOI:https://doi.org/10.1002/jhet.2552.
  • Navnath D. Rode, Amol D. Sonawane, Laxman Nawale, Vijay Khedkar, Ramesh A. Joshi, Anjali P. Likhite, Dhiman Sarkar And Rohini Joshi, Synthesis, biological evaluation, and molecular docking studies of novel 3-aryl-5-(alkyl-thio)-1H-1,2,4-triazoles derivatives targetting Mycobacterium tuberculosis, Chemical Biology and Drug Design., 90, 1206 - 1214 (2017), DOI:https://doi.org/10.1111/cbdd.13040.
  • Mahendra B. Rao, Sambhaji T. Dhumal, Amarsinh R. Deshmukh, Laxman Nawale, Vijay Khedkar, Dhiman Sarkar And Ramrao A. Mane, New bithiazolyl hydrazones: Novel synthesis, charcterization and antitubercular evaluation, Bioorganic & Medicinal Chemistry Letters., 27, 288 - 294 (2017), DOI:https://doi.org/10.1016/j.bmcl.2016.11.056.
  • Pramod V. Chavan, Kapil S. Pandit, Uday V. Desai, Prakash P. Wadgaonkar, Laxman Nawale, Sujit Bhansali And Dhiman Sarkar, Click-chemistry-based multicomponent condensation approach for design and synthesis of spirochromene-tethered 1,2,3-triazoles as potential antitubercular agents, Research on Chemical Intermediates., 43, 5675 - 5690 (2017), DOI:https://doi.org/10.1007/s11164-017-2955-y.
  • Laxman Nawale, Parul Dubey, Bhushan Chaudhari, Dhiman Sarkar And Asmita Prabhune, Anti-proliferative effect of novel primary cetyl alcohol derived sophorolipids against human cervical cancer cells HeLa, PLOS One., 12, (2017), DOI:https://doi.org/10.1371/journal.pone.0174241.
  • Preeti Nigam Joshi, Sachin Agawane, Meghana C. Athalye, Vrushali Jadhav, Dhiman Sarkar And Rajiv Prakash, Multifunctional inulin tethered silver-graphene quantum dots nanotheranostic module for pancreatic cancer therapy, Materials Science and Engineering: C., 78, 1203 - 1211 (2017), DOI:https://doi.org/10.1016/j.msec.2017.03.176.
  • Mubarak H. Shah, Dnyaneshwar D. Subhedar, Firoz A. Kalam Khan, Jaiprakash N. Sangshetti, Laxman Nawale, Manisha Arkile, Dhiman Sarkar And Bapurao B. Shingate, Synthesis of Novel Triazole-incorporated Isatin Derivatives as Antifungal, Antitubercular, and Antioxidant Agents and Molecular Docking Study, Journal of Heterocyclic Chemistry., 54, 413 - 421 (2017), DOI:https://doi.org/10.1002/jhet.2598.
  • Yogita K. Abhale, Amit V. Sasane, Abhijit P. Chavan, Saddam Husen Shekh, Keshav K. Deshmukh, Sujit Bhansali, Laxman Nawale, Dhiman Sarkar And Pravin C. Mhaske, Synthesis and antimycobacterial screening of new thiazolyl-oxazole derivatives, European Journal of Medicinal Chemistry., 132, 333 - 340 (2017), DOI:https://doi.org/10.1016/j.ejmech.2017.03.065.
  • Dnyaneshwar D Subhedar, Mubarak H. Shaikh, Bapurao B. Shingate, Laxman Nawale, Dhiman Sarkar, Vijay Khedkar, Firoz A. Khan And Jaiprakash N. Sangshetti, Quinolidene-rhodanine conjugates: Facile synthesis and biological evaluation, European Journal of Medicinal Chemistry., 125, 385 - 399 (2017), DOI:https://doi.org/10.1016/j.ejmech.2016.09.059.
  • Jaisingh M. Divse, Santosh B. Mhaske, Chaitanya R. Charolkar, Duhita G. Sant, Santosh G. Tupe, Mukund V. Deshpande, Vijay M. Khedkar, Laxman U. Nawale, Dhiman Sarkar And Vandana S. Pore, Synthesis and biological evaluation of new fluconazole B-lactam conjugates linked via 1,2,3-triazole, New Journal of Chemistry., 41, 470 - 479 (2017), DOI:10.1039/C6NJ03117J.
  • Yeware AM, Shurpali KD And Athalye MC and Sarkar D , Superoxide Generation and Its Involvement in the Growth of Mycobacterium smegmatis, Front. Microbiol., 8:105, (2017), DOI:10.3389/fmicb.2017.00105.
  • Dnyaneshwar D. Subhedar, Mubarak H. Shaikh, Laxman Nawale, Dhiman Sarkar, Vijay M. Khedkar And Bapurao B. Shingate, Quinolidene Based Monocarbonyl Curcumin Analogues as Promising Antimycobacterial Agents: Synthesis and Molecular Docking Study, Bioorganic & Medicinal Chemistry Letters., , (2017), DOI:10.1016/j.bmcl. 2017.01.004.
  • Mahesh M. Pisal , Laxman U. Nawale , Manoj D. Patil , Sujit G. Bhansali , Jayant M. Gajbhiye , Dhiman Sarkar , Subhash P. Chavan , Hanumant B. Borate And *, Hybrids of thienopyrimidinones and thiouracils as anti-tubercular agents: SAR and docking studies, European Journal of Medicinal Chemistry., 127, 459 - 469 (2017), DOI:10.1016/j.ejmech.2017.01.009.
  • Amol D. Sonawane, Navnath D. Rode, Laxman Nawale, Rohini R. Joshi* , Ramesh A. Joshi, Anjali P. Likhite And Dhiman Sarkar*, Synthesis and biological evaluation of 1,2,4-triazole-3-thione and 1,3,4-oxadiazole-2-thione as anti-mycobacterial agents, Chemical Biology & Drug Design., , (2017), DOI:10.1111/cbdd.12939.
  • Tushar R. Valkute · Manisha Arkile · Dhiman Sarkar · Asish K. Bhattacharya, Naturally Occurring Anti-TB Agents: Isolation, Chemical Transformations and In Vitro Antitubercular Activities of Secondary Metabolites of Rhizomes of Alpinia galanga, Planta Medica., , (2016), DOI:10.1055/s-0042-112226.
  • Mahendra B. Bhalerao, Sambhaji T. Dhumal, Amarsinh R. Deshmukh, Laxman U. Nawale, Vijay Khedkar, Dhiman Sarkar And Ramrao A. Mane, New bithiazolyl hydrazones: novel synthesis, characterization and antitubercular evaluation, Bioorganic & Medicinal Chemistry Letters., , (2016), DOI:http://dx.doi.org/10.1016/j.bmcl.2016.11.056.
  • Jaisingh M. Divse, Santosh B. Mhaske, Chitanya R. Charolkar, Duhita G Sant, Santosh G Tupe, Mukund V. Deshpande, vijay khedkar, Laxman Nawale And Dhiman Sarkar and Vandana Sudhir Pore, Synthesis and biological evaluation of new fluconazole ?-lactam conjugates linked via 1,2,3-triazole, New Journal of Chemistry., , (2016), DOI:10.1039/C6NJ03117J.
  • Dnyaneshwar D. Subhedar, Mubarak H. Shaikh, Bapurao B. Shingate, Laxman Nawale, Dhiman Sarkar, Vijay M. Khedkar, Firoz A. Kalam Khan And Jaiprakash N. Sangshetti, Quinolidene-rhodanine conjugates: Facile synthesis and biological evaluation, European Journal of Medicinal Chemistry., , (2016), DOI:10.1016/j.ejmech.2016.09.059.
  • Pal S, Ramu V, Taye N, Mogare DG, Yeware AM, Sarkar D, Reddy DS, Chattopadhyay And Das A, GSH Induced Controlled Release of Levofloxacin form a Pur-pose-built Prodrug: Luminescence Response for Probing the Drug Release in E-coli and Staphylococcus aureus, Bioconjugate Chemistry., , (2016), DOI:10.1021/acs.bioconjchem.6b00324.
  • Dnyaneshwar D. Subhedar, Mubarak H. Shaikh, Bapurao B. Shingate, Laxman Nawale And Dhiman Sarkar and Vijay M. Khedkar, Novel tetrazoloquinoline–thiazolidinone conjugates as possible antitubercular agents: synthesis and molecular docking, Med. Chem. Commun., , (2016), DOI:10.1039/C6MD00278A.
  • Pradip K. Gadekar, Abhijit Roychowdhury, Prashant S. Kharkar, Vijay Khedkar, Manisha Arkile, Hardik Manek, Dhiman Sarkar, Rajiv Sharma, V. Vijayakumar And S. Sarveswari, Design, synthesis and biological evaluation of novel azaspiro analogs of linezolid as antibacterial and antitubercular agents, European Journal of Medicinal Chemistry., , (2016), DOI:10.1016/j.ejmech.2016.07.001.
  • Pravin S. Mahajan†, Mukesh D. Nikam†, Laxman U. Nawale‡, Vijay M. Khedkar‡, Dhiman Sarkar‡ And and Charansingh H. Gill*†, Synthesis and Anti-tubercular Activity of New Benzo[b]thiophenes, ACS Med. Chem. Lett., , (2016), DOI:10.1021/acsmedchemlett.6b00077.
  • Subhedar DD , Shaikh MH , Arkile MA , Yeware A , Sarkar D And Shingate BB, Facile Synthesis of 1,3-Tiazolidin-4-ones as Antitubercular Agents, ChemInform., , 1704 - 1708 (2016), DOI:10.1002/chin.201629163.
  • Ruby Singh , Laxman Nawale , Dhiman Sarkar , C. G. Suresh (Contributed equally to this work: Ruby Singh And Laxman Nawale)., Two Chitotriose-Specific Lectins Show Anti- Angiogenesis, Induces Caspase-9-Mediated Apoptosis and Early Arrest of Pancreatic Tumor Cell Cycle, PLoS ONE., , (2016), DOI:http://dx.doi.org/10.1371/journal.pone.0146110.
  • Mubarak H. Shaikh · Dnyaneshwar D. Subhedar · Manisha Arkile · Vijay M. Khedkar · Nandadeep Jadhav · Dhiman Sarkar · Bapurao B. Shingate, Synthesis and bioactivity of novel triazole incorporated benzothiazinone derivatives as antitubercular and antioxidant agent, Bioorganic & Medicinal Chemistry Letters., 26, 561 - 569 (2016), DOI:doi:10.1016/j.bmcl.2015.11.071.
  • Mubarak H. Shaikh · Dnyaneshwar D. Subhedar · Firoz A. Kalam Khan · Jaiprakash N. Sangshetti · Laxman Nawale · Manisha Arkile · Dhiman Sarkar · Bapurao B. Shingate, Synthesis of Novel Triazole-incorporated Isatin Derivatives as Antifungal, Antitubercular, and Antioxidant Agents and Molecular Docking Study, Journal of Heterocyclic Chemistry., 9999, (2016), DOI:10.1002/jhet.2598.
  • Mubarak H. Shaikh, Bapurao B. Shingat, Laxman Nawale, Govinda R. Navale And Sandip S. Shinde, Synthesis, biological evaluation and molecular docking of novel coumarin incorporated triazoles as antitubercular, antioxidant and antimicrobial agents, Medicinal Chemistry Research., 25, 790 - 804 (2016), DOI:10.1007/s00044-016-1519-9.
  • Tabasum Ismail · Syed Shafi · Jada Srinivas · Dhiman Sarkar · Yasrib Qurishi · Jabeena Khazir · Mohammad Sarwar Alam · Halmuthur Mahabalarao Sampath Kumar, Synthesis and Tyrosinase Inhibition activity of trans-Stilbene Derivatives, Bioorganic Chemistry., 64, 97 - 102 (2016), DOI:10.1016/j.bioorg.2016.01.001.
  • Dnyaneshwar D. Subhedar · Mubarak H. Shaikh · Manisha A. Arkile · Amar Yeware · Dhiman Sarkar · Bapurao B. Shingate, Facile Synthesis of 1,3-Thiazolidin-4-ones as Antitubercular Agents, Bioorganic & Medicinal Chemistry Letters., 26, 1704 - 1708 (2016), DOI:10.1016/j.bmcl.2016.02.056.
  • N.C. Desai · Hardik Somani · Amit Trivedi · Kandarp Bhatt · Laxman Nawale · Vijay M. Khedkar · Prakash C. Jha · Dhiman Sarkar, Synthesis, biological evaluation and mo lecular docking study of some novel indole and pyridine based 1,3,4-oxadiaz ole derivatives as potential antituber- cular agents, Bioorganic & Medicinal Chemistry Letters., 26, 1776 - 1783 (2016), DOI:10.1016/j.bmcl.2016.02.043.
  • Priyanka R. Sharma · Sunil Kamble · Dhiman Sarkar · Amitesh Anand · Anjani J. Varma, Shape and size engineered cellulosic nanomaterials as broad spectrum anti-microbial compounds, nternational Journal of Biological Macromolecules., 87, 460 - 465 (2016), DOI:10.1016/j.ijbiomac.2016.02.024.
  • Varsha S. Honmorea, Supada R. Rojatkarb, Laxman U. Nawalec, Manisha A. Arkilec, Vijay M. Khedkarc, Arun D. Natua And Dhiman Sarkarc, In vitro and ex vivo antitubercular activity of diarylheptanoids from the rhizomes of Alpinia officinarum Hance, Natural Product Research., , (2016), DOI:10.1080/14786419.2016.1149702.
  • Dnyaneshwar D. Subhedar · Mubarak H. Shaikh · Laxman Nawale · Amar Yeware · Dhiman Sarkar · Bapurao B. Shingate, [Et3NH][HSO4] catalyzed efficient synthesis of 5-arylidene-rhodanine conjugates and their antitubercular activity, Research on Chemical Intermediates., , (2016), DOI:10.1007/s11164-016-2484-0.
  • Dnyaneshwar D. Subhedara, Mubarak H. Shaikha, Laxman Nawaleb, Amar Yewareb, Dhiman Sarkarb, Firoz A. Kalam Khanc, Jaiprakash N. Sangshettic, Bapurao B. Shingatea, And , Novel Tetrazoloquinoline-Rhodanine Conjugates: Highly Efficient Synthesis and Biological Evaluation, Bioorganic & Medicinal Chemistry Letters., 26, 2278 - 2283 (2016), DOI:doi:10.1016/j.bmcl.2016.03.045.
  • Ashish A. Chinchansure1, Manisha Arkile2, Dinesh R. Shinde3, Dhiman Sarkar2 And Swati P. Joshi1, A New Dinor-cis-Labdane Diterpene and Flavonoids with Antimycobacterium Activity from Colebrookea oppositifolia, Planta Medica Letters., , (2016), DOI:10.1055/s-0042-102200.
  • Chitre TS1, Asgaonkar KD2, Miniyar PB3, Dharme AB2, Arkile MA4, Yeware A4, Sarkar D4, Khedkar VM5 And Jha PC6., Synthesis and docking studies of pyrazine-thiazolidinone hybrid scaffold targeting dormant tuberculosis, Bioorganic & Medicinal Chemistry Letters., 26, 2224 - 2228 (2016), DOI:doi:10.1016/j.bmcl.2016.03.055.
  • Honmore VS1, Kandhare AD2, Kadam PP2, Khedkar VM3, Sarkar D3, Bodhankar SL4, Zanwar AA5, Rojatkar SR6 And Natu AD7, Isolates of Alpinia officinarum Hance as COX-2 inhibitors: Evidence from anti-inflammatory, antioxidant and molecular docking studies, International Immunopharmacology., 33, 8 - 17 (2016), DOI:doi:10.1016/j.intimp.2016.01.024.
  • Singh R, Nawale L, Arkile M, Wadhwani S, Shedbalkar U, Chopade S, Sarkar D And Chopade BA, Phytogenic silver, gold, and bimetallic nanoparticles as novel antitubercular agents, International Journal of Nanomedicine., Volume 11, 1889 - 1897 (2016), DOI:https://dx.doi.org/10.2147/IJN.S102488.
  • Sambhaji T. Dhumal · Amarsinh R. Deshmukh · Manisha R. Bhosle · Vijay M. Khedkar · Laxman U. Nawale · Dhiman Sarkar · Ramrao A. Mane, Synthesis and Antitubercular Activity of New 1,3,4-Oxadiazoles Bearing Pyridyl and Thiazolyl Scaffolds, Bioorganic & Medicinal Chemistry Letters., , (2016), DOI:http://dx.doi.org/10.1016/j.bmcl.2016.05.093.
  • Sambhaji T. Dhumal · Amarsinh R. Deshmukh · Manisha R. Bhosle · Vijay M. Khedkar · Laxman U. Nawale · Dhiman Sarkar · Ramrao A. Mane, Synthesis and Antitubercular Activity of New 1,3,4-Oxadiazoles Bearing Pyridyl and Thiazolyl Scaffolds, Bioorganic & Medicinal Chemistry Letters., , (2016), DOI:http://dx.doi.org/10.1016/j.bmcl.2016.05.093.
  • Laxman Nawale · Dhiman Sarkar, Efficacy Study Of Potential Anti-tubercular Molecules: In-vitro and Ex-vivo, Conference Paper., , (2015).
  • Laxman Nawale · Dhiman Sarkar, A QUANTITATIVE, AUTOMATED, HIGH CONTENT SCREENING ASSAY APPROACH TO ANTI-ANGIOGENICDRUG DISCOVERY, Conference Paper., , (2015).
  • Laxman Nawale · Dhiman Sarkar, Discovery of new chemical entities against diseases of national importance :an HTS approach, Conference Paper., , (2015).
  • Vivek Khilari · Laxman Nawale · Dhiman Sarkar · Bhaskar Idage · Susheela Idage, BIODRGRADABLE CHITOSAN GRAFT POLY(LACTIC ACID) NANOPARTICLES AS NANOCARRIERS FOR ANTI-TB DRUG (ISONIAZID), Conference Paper., , (2015).
  • Parul Dubeya · Laxman Nawaleb · Dhiman Sarkarb · Anuya Nisalc · Asmita Prabhunea, Mechanistic understanding of rapid gelation of Silk fibroin using a biosurfactant – Sophorolipid, Conference Paper., , (2015).
  • Ruby Singha · Laxman Nawaleb · Sushama M. Gaikwada · Dhiman Sarkarb · C.G. Suresha, Purification and characterization of an agglutinin from Datura innoxia with antineoplastic activity, Conference Paper., , (2015).
  • Laxman Nawale · Hardik Manek · Nandadeep Jadhav · Jennifer Cheruvathur · Dhiman Sarkar, High Throughput Screening of Inhibitors for Tuberculosis at NCL : A Novel Drug Discovery Initiative from CSIR, Conference Paper., , (2015).
  • Preeti Nigam · Dhiman Sarkar, Multifunctional Silica Nanoparticles for Pancreatic Cancer Specific Drug Delivery and Bioimaging, Journal ofChemistry & Applied Biochemistry., 2, (2015).
  • Shamim Akhtar · Sheetal Singh · Santosh Kumar · Dhiman Sarkar, Analyzing Different Acetyl Co-A Metabolizing Enzymes as Potential Drug Targets against Mycobacterium tuberculosis, British Microbiology Research Journal., 10, (2015), DOI:10.9734/BMRJ/2015/19032.
  • Sambhaji T. Dhumal · Amarsinh R. Deshmukh · Lalit D. Khillare · Manisha Arkile · Dhiman Sarkar · and Ramrao A. Mane, Synthesis and Antitubercular activity of New Thiazolidinones with Pyrazinyl and Thiazolyl scaffolds, Journal of Heterocyclic Chemistry., , (2015), DOI:10.1002/jhet.2552.
  • Madhukar S Said · Ashish A Chinchansure · Laxman Nawale · Ankita Durge · Ashish Wadhwani · Smita S Kulkarni · Dhiman Sarkar · Swati · P Joshi, A new butenolide cinnamate and other biological active chemical constituents from Polygonum glabrum, Natural product research., 29(22), 2080 - 6 (2015), DOI:10.1080/14786419.2015.1004674.
  • Parul Dubey · Laxman Nawale · Dhiman Sarkar · Anuya Nisal · Asmita A Prabhune, Sophorolipid assisted tunable and rapid gelation of silk fibroin to form porous biomedical scaffolds, RSC Advances., 5, 33955 - 33962 (2015), DOI:10.1039/C5RA04317D.
  • Abhishek Mishra · Dhiman Sarkar, Qualitative and quantitative proteomic analysis of Vitamin C induced changes in Mycobacterium smegmatis, Frontiers in Microbiology., 6, 451 (2015), DOI:10.3389/fmicb.2015.00451.
  • Richa Singh · Laxman U Nawale · Manisha Arkile · Utkarsha U Shedbalkar · Sweety A Wadhwani · Dhiman Sarkar · Balu A Chopade, Chemical and biological metal nanoparticles as antimycobacterial agents: A comparative study, International Journal of Antimicrobial Agents., 46(2), 183 - 8 (2015), DOI:10.1016/j.ijantimicag.2015.03.014.
  • Mubarak H. Shaikh · Dnyaneshwar D. Subhedar · Laxman Nawale · Dhiman Sarkar · Firoz A. Kalam Khan · Jaiprakash N. Sangshetti · Bapurao B. Shingate, 1,2,3-Triazole derivatives as antitubercular agents: synthesis, biological evaluation and molecular docking study, Medicinal Chemistry Communication., 6, 1104 - 1116 (2015), DOI:10.1039/c5md00057b.
  • Roshan R Kulkarni · Ketaki Shurpali · Vijay M Khedkar · Vedavati G Puranik · Dhiman Sarkar · Swati P Joshi, New pimarane diterpenes and other antimycobacterial metabolites from Anisochilus verticillatus, Natural product research., 30(6), 675 - 681 (2015), DOI:10.1080/14786419.2015.1040990.
  • Nilesh R Tawari · Seema Bag · Archana Raju · Arundhati C Lele · Ranjeet Bairwa · Mukti Kanta Ray · Mgr Rajan · Laxman U Nawale · Dhiman Sarkar · Mariam S Degani, Rational drug design, synthesis and biological evaluation of dihydrofolate reductase inhibitors as antituberculosis agents, Future medicinal chemistry., 7(8), 979 - 88 (2015), DOI:10.4155/fmc.15.48.
  • Rima Bharadwaj · Ashish A. Chinchansure · Roshan R. Kulkarni · Manisha Arkile · Dhiman Sarkar · Swati P. Joshi, Rottlerin Derivatives and Other Compounds from Mallotus philippinensis Fruits and Their Potential Antimycobactrial Activity, Planta Medica Letters., 2, 28 - 30 (2015), DOI:10.1055/s-0035-1557793.
  • Ashish Chinchansure · Manisha Arkile · Anurag Shukla · Shanmugam Dhanasekaran · Dhiman Sarkar · Swati P. Joshi, Leucas mollissima, a Source of Bioactive Compounds with Antimalarial and Antimycobacterium Activities, Planta Medica Letters., 2, 35 - 38 (2015), DOI:10.1055/s-0035-1557830.
  • Sarvesh K Soni · Sampa Sarkar · Selvakannan R. Periasamy · Dhiman Sarkar · Suresh K Bhargava, Intrinsic therapeutic and biocatalytic roles of ionic liquid mediated self-assembled platinum-phytase nanosphere, RSC Advances., 5, 62871 - 62881 (2015), DOI:10.1039/c5ra11273g.
  • Pravin S. Mahajan · Mukesh D. Nikam · Vijay M. Khedkar · Prakash C. Jha · Dhiman Sarkar · Charansingh H. Gill, Synthesis, biological evaluation and molecular docking studies of N-acylheteroaryl hydrazone derivatives as antioxidant and anti-inflammatory agents, Research on Chemical Intermediates., , (2015), DOI:10.1007/s11164-015-2176-1.
  • Ashish Chinchansure · Neelam Shamnani · Manisha Arkile · Dhiman Sarkar · Swati Joshi, ANTIMYCOBACTERIUM ACTIVITY OF COUMARINS FROM FRUIT PULP OF AEGLE MARMELOS (L.) CORREA, International Journal of Basic and Applied Chemical Sciences., 5, 39 - 44 (2015).
  • Vandana S. Pore, Jaisingh M. Divse, Chaitanya R. Charolkar, Laxman U. Nawale, Vijay M. Khedkar And Dhiman Sarkar, Design and synthesis of 11? - substituted bile acid derivatives as potential anti - tuberculosis agents, Bioorganic & Medicinal Chemistry Letters., 25, 4185 - 4190 (2015), DOI:10.1016/j.bmcl.2015.08.006.
  • Arundhati C. Lele · Archana Raju · Mihir P. Khambete · M. K. Ray · M. G. R. Rajan · Manisha A. Arkile · Nandadeep J. Jadhav · Dhiman Sarkar · Mariam S. Degan, Design and Synthesis of a Focused Library of Diamino Triazines as Potential Mycobacterium tuberculosis DHFR Inhibitors, ACS Med Chem Lett., 6 (11), 1140 - 1144 (2015), DOI:10.1021/acsmedchemlett.5b00367.
  • Hanumant Bapurao Borate · Ritesh A. Annadate · Sandip S. Vagh · Mahesh M. Pisal · Sagar B. Deokate · Manisha A. Arkile · Nandadeep J. Jadhav · Laxman U. Nawale · Dhiman Sarkar, Synthesis and evaluation of thieno[2,3-d]pyrimidin-4(3H)-ones as potential antitubercular agents, Medicinal Chemistry Communication., , (2015), DOI:10.1039/C5MD90062J.
  • Preeti Nigam · Shobha Waghmode · Michelle Louis · Shishanka Wangnoo · Pooja Chavan · Dhiman Sarkar, Materials Chemistry B, Journal of Materials Chemistry., , (2014), DOI:10.1039/c4tb00015c.
  • Rohit R Joshi · Avinash Barchha · Vijay M Khedkar · Raghuvir R S Pissurlenkar · Sampa Sarkar · Dhiman Sarkar · Rohini R Joshi · Ramesh A Joshi · Anamik K Shah · Evans C Coutinho, Targeting Dormant Tuberculosis Bacilli: Results for Molecules with a Novel Pyrimidone Scaffold, Chemical Biology & Drug Design., 85(2), 201 - 207 (2014), DOI:10.1111/cbdd.12373.
  • Ketaki Dilip Shurpali · Upasana Singh · Shamim Akhtar Sampa Sarkar · Abhishek Mishra · Roshan Kulkarni · Swati Joshi · Dhiman Sarkar, Advanced cell-based high-throughput screening assays targeting active and latent Mycobacterium tuberculosis, Journal of Biotechnology., 185, S18 (2014), DOI:10.1016/j.jbiotec.2014.07.061.
  • Preeti Nigam · Shobha Waghmode · Amar Yeware · Laxman Nawale · Priyanka Dagde · Amol Dhudhane · Dhiman Sarkar, Aptamer Functionalized Multifunctional Fluorescent Nanotheranostic Platform for Pancreatic Cancer, Journal of Nanopharmaceutics and Drug Delivery., 2, 280 - 287 (2014), DOI:10.1166/jnd.2014.1070.
  • Roshan R. Kulkarni, Santosh G. Tupe, Suwarna P. Gample, Macchindra G. Chandgudea, Dhiman Sarkar And Mukund V. Deshpande & Swati P. Joshi, Antifungal dimeric chalcone derivative kamalachalcone E from Mallotus philippinensis, Natural Product Research., 28, 245 - 250 (2014), DOI:10.1080/14786419.2013.843178.
  • Shamim Akhtar · Arshad Khan · Charles D Sohaskey · Chinnaswamy Jagannath · Dhiman Sarkar, Nitrite Reductase NirBD Is Induced and Plays an Important Role during In Vitro Dormancy of Mycobacterium tuberculosis, Journal of bacteriology., 195, 4592 - 4599 (2013), DOI:10.1128/JB.00698-13.
  • Roshan R Kulkarni · Ketaki Shurpali · Vedavati G Puranik · Dhiman Sarkar · Swati P Joshi, Antimycobacterial Labdane Diterpenes from Leucas stelligera, J Nat Prod., 76, 1836 - 1841 (2013), DOI:10.1021/np400002p.
  • Roshan R Kulkarni · Santosh G Tupe · Suwarna P Gample · Macchindra G Chandgude · Dhiman Sarkar · Mukund V Deshpande · Swati P Joshi, Antifungal dimeric chalcone derivative kamalachalcone E from Mallotus philippinensis, Natural product research., 28, 245 - 250 (2013), DOI:10.1080/14786419.2013.843178.
  • Shafeek A. R. Mulla · Mohsinkhan Y. Pathan · Santosh S. Chavan · Suwara P. Gample · Dhiman Sarkar, Highly efficient one-pot multi-component synthesis of a-aminophosphonates and bis-a- aminophosphonates catalyzed by heterogeneous reusable silica supported dodecatungstophosphoric acid (DTP/SiO2) at ambient temperature and their antitubercular evaluation against Mycobactrium Tuberculosis, RSC Advances., 4, 7666 - 7672 (2013), DOI:10.1039/C3RA45853A.
  • Rohan A. Limaye, Virendra B. Kumbhar, Arun D. Natu, Madhusudan V. Paradkar, Varsha S. Honmore, Rubia R. Chauhan, Suwarna P. Gample And Dhiman Sarkar, One pot solvent free synthesis and in vitro antitubercular screening of 3-Aracylphthalides against Mycobacterium tuberculosis, Bioorganic & Medicinal Chemistry Letters., 23, 711 - 714 (2013), DOI:10.1016/j.bmcl.2012.11.097.
  • Roshan R. Kulkarni, Ketaki Shurpali, Vedavati G. Puranik And Dhiman Sarkar and Swati P. Joshi, Antimycobacterial Labdane Diterpenes from Leucas stelligera, Journal of Natural Products., 76 (10), 1836 - 1841 (2013).
  • Shamim Akhtar, Arshad Khan, Charles D. Sohaskey And Chinnaswamy Jagannath and Dhiman Sarkar, Nitrite Reductase NirBD is induced and plays and important role during in vivo dormancy of Mycobacterium tuberculosis, Journal of Bacteriology., vol. 195 no. 20, 4592 - 4599 (2013).
  • R. R. Kulkarni · K. D. Shurpali · R. I. Gawde · D. Sarkar · V. G. Puranik · S. P. Joshi, Chemical investigation of Plectranthus mollis, Journal of Medicinal and Aromatic Plant Sciences., , (2012).
  • Roshan R Kulkarni · Ketaki Shurpali · Rupesh L Gawde · Dhiman Sarkar · Vedavati G Puranik · Swati P Joshi, Phyllocladane diterpenes from Anisomeles heyneana, Journal of Asian natural products research., , (2012).
  • Rohan A Limaye · Virendra B Kumbhar · Arun D Natu · Madhusudan V Paradkar · Varsha S Honmore · Rubia R Chauhan · Suwarna P Gample · Dhiman Sarkar, ChemInform Abstract: One Pot Solvent Free Synthesis and in vitro Antitubercular Screening of 3-Aracylphthalides Against Mycobacterium tuberculosis, Bioorganic & Medicinal Chemistry Letters., , (2012), DOI:10.1002/chin.201321107.
  • Sampa Sarkar And Dhiman Sarkar, Potential use of nitrate reductase as a biomarker for the identification of active and dormant inhibitors of Mycobacterium tuberculosis in a THP-1 infection model, Journal of Biomolecular Screening., vol. 17 no. 7, 966 - 973 (2012).
  • Upasana Singh · Shamim Akhtar · Abhishek Mishra · Dhiman Sarkar, A novel screening method based on menadione mediated rapid reduction of tetrazolium salt for testing of anti-mycobacterial agents, Journal of microbiological methods., 84, 202 - 207 (2011), DOI:10.1016/j.mimet.2010.11.013.
  • Arshad Khan · Dhiman Sarkar, Nitrate reduction pathways in mycobacteria and their implications during latency, Microbiology., 158, 301 - 307 (2011), DOI:10.1099/mic.0.054759-0.
  • Sarvesh K Soni · Sampa Sarkar · Dhiman Sarkar · Peter J Coloe · Suresh K Bhargava · Vipul Bansal, SELF–ASSEMBLED HISTIDINE ACID PHOSPHATE NANOCAPSULES AS TEMPLATES FOR MULTIFUNCTIONAL HOLLOW PLATINUM NANOSPHERES IN IONIC LIQUID [BMIM][BF 4 ] FOR DRUG DELIVERY, Proceedings of Chemeca., , (2011).
  • Shamim Akhtar, Sampa Sarkar, Abhishek Mishra And Dhiman Sarkar, A method to extract intact and pure RNA from mycobacteria, Analytical Biochemistry., 417(2), 286 - 288 (2011).
  • Dasari Sreekanth · Asad Syed · Sampa Sarkar · Dhiman Sarkar · B Santhakumari · Absar Ahmad · Islam Khan, Production, purification and characterization of taxol and 10DAB III from a new endophytic fungus Gliocladium sp. isolated from the Indian yew tree, Taxus baccata, Journal of Microbiology and Biotechnology., 19, 1342 - 1347 (2009).
  • Arshad Khan · Shamim Akhtar · Jawid N Ahmad · Dhiman Sarkar, Presence of a functional nitrate assimilation pathway in Mycobacterium smegmatis, Microbial Pathogenesis., 44, 71 - 77 (2008).
  • A. Khan, S. Sarkar And D. Sarkar, Bactericidal activity of 2-nitroimidazole against the active replicating stage of Mycobacterium bovis BCG and Mycobacterium tuberculosis with intracellular efficacy in THP-1 macrophages, Int. J Antimicrob Agents., 32(1), 40 - 45 (2008).
  • A. Khan And D. Sarkar, A simple whole cell based high throughput screening protocol using Mycobacterium bovis BCG for inhibitors against dormant and active tubercle bacilli, Microbiol Methods., 73(1), 62 - 68 (2008).
  • A. Khan, S. Akhtar, J N Ahmad And D Sarkar, Presence of functional nitrate assimilation pathway in Mycobacterium smegmatis, . Jan; 44(1):71-7, Microb Pathog., 44, 71 - 77 (2008).
  • A Khan And D Sarkar, Identification of a respiratory-type nitrate reductase and its role for survival of Mycobacterium smegmatis in Wayne model, Microb Pathog., 41(2-3), 90 - 95 (2006).
  • U Singh And D Sarkar, Development of a simple high-throughput screening protocol based on biosynthetic activity of Mycobacterium tuberculosis glutamine synthetase for the identification of novel inhibitors, J Biomolecular Screening., 11(8), 1035 - 1042 (2006).
  • J Bhat, R Rane, S M Solapure, D Sarkar, U Sharma, M N Harish, S Lamb, D Plant, P Alcock, S Peters, S Barde And R K Roy, High-throughput screening of RNA polymerase inhibitors using a fluorescent UTP analog, J. Biomol. Screen., 11(8), 968 - 976 (2006).
  • Upasana Singh · Vinita Panchanadikar · Dhiman Sarkar, Development of a Simple Assay Protocol for High-Throughput Screening of Mycobacterium tuberculosis Glutamine Synthetase for the Identification of Novel Inhibitors, Journal of Biomolecular Screening., 10, 725 - 729 (2005).
  • U Singh, V Panchanadikar And D Sarkar, Development of a simple assay protocol for high-throughput screening of Mycobacterium tuberculosis glutamine synthetase for the identification of novel inhibitors, J Biolecular Screening., 10(7), 725 - 729 (2005).
  • D Sarkar, I Ghosh And S Datta, Biochemical characterization of Plasmodium falciparum hypoxanthine-guanine-xanthine phosphorbosyltransferase: role of histidine residue in substrate selectivity, Mol Biochem Parasitol., 137(2), 267 - 276 (2004).
  • D. Sarkar and A. Bhaduri, Temperature induced rapid rise in cytoplasmic free Ca2+ concentration in pathogenic Leishmania donovani promastigotes, FEBS letters., 375, 83 - 86 (1995).
  • Dhiman Sarkar · Anil Ghosh · Amarnath Bhaduri, Possible involvement of Ca2+ in the in vitro morphogenetic transformation of Leishmania donovani amastigotes to promastigotes, Proceedings of the Indian National Science Academy. Part B Biological sciences., 58, 281 - 288 (1992).
  • M. Ray, D. Sarkar And S. Ray, Aminoacetone synthase from goat liver involvement of arginine residue at the active site and on the stability of the enzyme, J Biochem., 275, 575 - 579 (1991).