Research Group Publications
 
  • Lakshmi Goswami‡, Lovely Gupta‡, Sayantan Paul, Maansi Vermani And Pooja Vijayaraghavan* and Asish K. Bhattacharya*, Design and synthesis of eugenol/isoeugenol glycoconjugates and other analogues as antifungal agents against Aspergillus fumigatus†, RSC Med. Chem., , (2022), DOI:DOI: 10.1039/D2MD00138A.
  • Lovely Gupta, Pooja Sen, Asish K. Bhattacharya And Pooja Vijayaraghavan, Isoeugenol affects expression pattern of conidial hydrophobin gene RodA and transcriptional regulators MedA and SomA responsible for adherence and biofilm formation in Aspergillus fumigatus, Archives of Microbiology (Springer)., 204:214, 1 - 14 (2022), DOI:https://doi.org/10.1007/s00203-022-02817-w.
  • Eswar K. Aratikatla, Md Kalamuddin, Kalpeshkumar C. Rana, Gaurav Datta, Mohd Asad, Srividhya Sundararaman, Pawan Malhotra, Asif Mohmmed And Asish K. Bhattacharya, Combating multi-drug resistant malaria parasite by inhibiting falcipain-2 and heme-polymerization: Artemisinin-peptidyl vinyl phosphonate hybrid molecules as new antimalarials, European Journal of Medicinal Chemistry., 220, (2021), DOI:https://doi.org/10.1016/j.ejmech.2021.113454.
  • Tharun K. Kotammagari, Sayantan Paul, Ganesh K. Barik And Manas K. Santra and Asish K. Bhattacharya, Synthesis of artemisinic acid derived glycoconjugates and their anticancer studies, Organic & Biomolecular Chemistry., , 1 - 13 (2020), DOI:DOI: 10.1039/D0OB00216J.
  • Eswar K. Aratikatla, Md Kalamuddin, Pawan Malhotra, Asif Mohmmed And * and Asish K. Bhattacharya*, Enantioselective Synthesis of ??Phenyl-?-amino Vinyl Phosphonates and Sulfones and Their Application to the Synthesis of Novel Highly Potent Antimalarials, ACS Omega., 5, 29025 - 29037 (2020), DOI:https://dx.doi.org/10.1021/acsomega.0c03470.
  • Tharun K. Kotammagari And Sayantan Paul and Asish K. Bhattacharya, Unusual Epimerization in Styryllactones: Synthesis of (?)-5- Hydroxygoniothalamin, (?)-5-Acetylgoniothalamin, and O?TBSGoniopypyrone, ACS Omega., 4, 22549 - 22556 (2019), DOI:DOI: 10.1021/acsomega.9b03263.
  • Sachin B. Agawane, Vidya S. Gupta, Mahesh J. Kulkarni, Asish K. Bhattacharya And Santosh S. Koratkar, Chemo-biological evaluation of antidiabetic activity of Mentha arvensis L. and its role in inhibition of advanced glycation end products, Journal of Ayurveda and Integrative Medicine., 10, 166 - 170 (2019), DOI:http://dx.doi.org/10.1016/j.jaim.2017.07.003.
  • Sachin B. Agawane, Vidya S. Gupta, Mahesh J. Kulkarni, Asish K. Bhattacharya, Santosh S. Koratkar And Vamkudoth Koteswara Rao, Patho-physiological evaluation of Duranta erecta for the treatment of urolithiasis, Journal of Ayurveda and Integrative Medicine., 10, 4 - 11 (2019), DOI:http://dx.doi.org/10.1016/j.jaim.2017.08.001.
  • Eswar K Aratikatla And and Asish K. Bhattacharya, A Short Review on Synthetic Routes of Antiepileptic Drug (R)-Lacosamide, Org. Process Res. Dev., , 1 - 20 (2019), DOI:DOI: 10.1021/acs.oprd.9b00373.
  • Hemender R. Chand and Asish K. Bhattacharya, Hemiketal-Keto Tautomerism in 2-Deoxy-?-lactones Mediated by 2-Lithiothiazole in Solution State: A Formal Synthesis of DAH, Kamusol and Their C5 Epimers, Asian J. Org. Chem., 8, 2113 - 2120 (2019), DOI:DOI: 10.1002/ajoc.201900407.
  • L. Goswami, S. Paul. T. K. Kotammagari And A. K. Bhattacharya*, Synthesis of artemisinin derived glycoconjugates inspired by click chemistry, New J. Chem., 43, 4017 - 4021 (2019).
  • T. R. Valkute, E. K. Aratikatla, N. Gupta, S. Ganga, M. K. Santra And A. K. Bhattacharya*, Synthesis and anticancer studies of Michael adducts and Heck arylation products of sesquiterpene lactones, zaluzanin D and zaluzanin C from Vernonia arborea, RSC Advances., 8, 38289 - 38304 (2018).
  • S. Paul And A. K. Bhattacharya*, Hydroxyl directed C-arylation: synthesis of 3-hydroxyflavones and 2-phenyl-3-hydroxy pyran-4-ones under transition-metal free conditions, Org. Biomol. Chem., 16, 444 - 451 (2018).
  • T. K. Kotammagari, R. G. Gonnade And A. K. Bhattacharya*, Biomimetic total synthesis of angiopterlactone B and other potential natural products, Org. Lett., 19(13), 3564 - 3567 (2017).
  • E. K. Aratikatla, T. R. Valkute, S. K. Puri, K. Srivastava And A. K. Bhattacharya*, Norepinephrine alkaloids as antiplasmodial agents: Synthesis of syncarpamide and insight into the structure-activity relationships of its analogues as antiplasmodial agents, Eur. J. Med. Chem., 138, 1089 - 1105 (2017).
  • T. R. Valkute, E. K. Aratikatla And A. K. Bhattacharya*, Efficient synthesis of functionalized olefins by Wittig reaction using Amberlite resin as a mild base, Synth. Commun., 47, 581 - 589 (2017).
  • H. R. Chand And A. K. Bhattacharya*, Diastereoselective synthesis of ?-ether derivatives of artemisinin, an antimalarial drug: The effect of nitrile on stereoselectivity, Asian J. Org. Chem., 5(2), 5802 - 5803 (2016).
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  • T. R. Valkute, M. Arkile, D. Sarkar And A. K. Bhattacharya.*, Naturally occurring anti-TB agents: isolation and in vitro antitubercular activities of secondary metabolites of rhizomes of Alpinia galanga, Planta Medica Int. Open., 3(3), e55 - e59 (2016).
  • T. K. Kotammagari, R. G. Gonnade And A. K. Bhattacharya*, Synthesis of naturally occurring (+)-osmundalactone and 4-epi-(+)-osmundalactone from triacetyl-O-D-glucal, Tetrahedron Lett., 56, 2783 - 2786 (2015).
  • A. K. Bhattacharya, * H. R. Chand, J. John And M. V. Deshpande, Clerodane type diterpene as a novel antifungal agent from Polyalthia longifolia var. pendula, Eur. J. Med. Chem., 94, 1 - 7 (2015).
  • I. K. Polanki, S. H. Kurma And A. K. Bhattacharya*, Direct glycosylation of unprotected and unactivated sugars using bismuth nitrate pentahydrate, J. Carbohydr. Chem., 34, 196 - 205 (2015).
  • E. K. Aratikatla And A. K. Bhattacharya*, Chiral pool approach for the synthesis of functionalized amino acids: Synthesis of antiepileptic drug (R)-Lacosamide, Tetrahedron Lett., 56, 5802 - 5803 (2015).
  • A. K. Bhattacharya, * S. S. Dange, I. K. Polanki And H. R. Chand, An efficient synthesis of 1,5-benzodiazepines catalyzed by bismuth nitrate, Ind. J. Chem., 53B, 1561 - 1567 (2014).
  • A. K. Bhattacharya, * D. S. Raut, K. C. Rana, I. K. Polanki, M. S. Khan And S. Iram, Diversity-oriented synthesis of ?-aminophosphonates: a new class of potential anticancer agents, Eur. J. Med. Chem., 66, 146 - 152 (2013).
  • A. K. Bhattacharya* And M. Mujahid, An efficient bakers’ yeast catalyzed multicomponent synthesis of ?-aminophosphonates in one-pot, Synth. Commun., 43, 2583 - 2589 (2013).
  • A. K. Bhattacharya* And K. C. Rana, Antimycobacterial agent, (E)-phytol and lauric amide from the plant Lagascea mollis, Ind. J. Chem., 52B, 901 - 903 (2013).
  • A. K. Bhattacharya, * K. C. Rana, C. Pannecouque And E. De Clercq, An efficient synthesis of a hydroxyethylamine (HEA) isostere and its ?-aminophosphonate and phosphoramidate derivatives as potential anti-HIV agent, ChemMedChem., 7, 1601 - 1611 (2012).
  • A. K. Bhattacharya, * K. C. Rana, D. S. Raut, V. P. Mhaindarkar And M. I. Khan, An efficient synthesis of benzodiazepinyl phosphonates as clostripain inhibitors via FeCl3 catalyzed four-component reaction, Org. Biomol. Chem., 9, 5407 - 5413 (2011).
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  • A. K. Bhattacharya* And K. C. Rana, Design, synthesis and biological evaluation of peptidyl-vinylaminophosphonates as novel cysteine protease inhibitors, Bioorg. Med. Chem., 19, 7129 - 7135 (2011).
  • A. K. Bhattacharya, * T. Kaur And K. N. Ganesh, Synthesis of the antibacterial benzoquinone primin and its water-soluble analogue, primin acid, Synthesis., , 1141 - 1144 (2010).
  • A. K. Bhattacharya, * K. C. Rana, M. Mujahid, I. Sehar And A. K. Saxena, Synthesis and in vitro study of 14-aryl-14H-dibenzo[a.j]xanthenes as cytotoxic agents, Bioorg. Med. Chem. Lett., 19, 5590 - 5593 (2009).
  • A. K. Bhattacharya, * M. Mujahid And A. A. Natu, An efficient method for the synthesis of acylals from aldehydes under solvent-free conditions catalysed by antimony trichloride, Synth. Commun., 38, 128 - 134 (2008).
  • A. K. Bhattacharya, * M. A. Diallo And K. N. Ganesh, SbCl3 as a highly efficient catalyst for the acetylation of alcohols, phenols and amines under solvent-free conditions, Synth. Commun., 38, 1518 - 1526 (2008).
  • A. K. Bhattacharya And * K. C. Rana, Amberlite-IR 120 catalyzed three-component synthesis of ?-amino phosphonates in one-pot, Tetrahedron Lett., 49(16), 2598 - 2601 (2008).
  • A. K. Bhattacharya, * A. K. Pathak And R. P. Sharma, Semi-synthesis of deoxyartemisinin, Mendeleev Commun., 17(1), 27 - 28 (2007).
  • A. K. Bhattacharya And * T. Kaur, An efficient one-pot synthesis of ?-amino phosphonates catalyzed by bismuth nitrate pentahydrate, Synlett., , 745 - 748 (2007).
  • A. K. Bhattacharya And * K. C. Rana, Microwave assisted synthesis of 14-aryl-14H-dibenzo[a.j]xanthenes catalysed by methanesulphonic acid under solvent-free condition, Mendeleev Commun., 17(4), 247 - 248 (2007).
  • Arvind S. Negi , Sunil K. Chattopadhyay And Sachin Srivastava & Asish K. Bhattacharya, A Simple Regioselective Demethylation of p?Aryl Methyl Ethers Using Aluminum Chloride?Dichloromethane System, Synthetic Communications., 35:1, 15 - 21 (2006), DOI:https://doi.org/10.1081/SCC-200046477.
  • Arvind Singh Negi, Mahinder P. Darokar, Sunil K. Chattopadhyay, Ankur Garg, Asish K. Bhattacharya And Vandana Srivastava and Suman P. S. Khanuja, Synthesis of a novel plant growth promoter from gallic acid, Bioorganic & Medicinal Chemistry Letters., 15, 1243 - 1247 (2005), DOI:doi:10.1016/j.bmcl.2004.11.079.
  • Sunil K. Chattopadhyay, * Sachin Srivastava, Koneni V. Sashidhara, Arun K. Tripathi And Asish K. Bhattacharya and Arvind S. Negi, Betuligenol derivative with growth inhibition and antifeedant activity, Bioorganic & Medicinal Chemistry Letters., 14, 1729 - 1731 (2004), DOI:doi:10.1016/j.bmcl.2004.01.040.
  • A. K. Bhattacharya, * M. Pal, D. C. Jain, B. S. Joshi, R. Roy, U. Rychlewska And R. P. Sharma, Stereoselective reduction of arteannuin B and its chemical transformations. A. K. Bhattacharya,* M. Pal, D. C. Jain, B. S. Joshi, R. Roy, U. Rychlewska and R. P. Sharma, Tetrahedron., 59(16), 2871 - 2876 (2003).
  • A. K. Bhattacharya, F. Stolz, J. Kurzeck, W. Rueger And R. R. Schmidt, SAR directed design and synthesis of novel ?(1-4)-glucosyltransferase inhibitors and their in vitro inhibition studies, Bioorg. Med. Chem., 10(4), 1129 - 1136 (2002).
  • A. K. Bhattacharya, F. Stolz, J. Kurzeck, W. Rueger And R. R. Schmidt, Structure-based design, synthesis and in vitro evaluation of substituted aryl/hetaryl methyl phosphonate and phosphate - UMP derivatives as potential glucosyltransferase inhibitors, Can. J. Chem., 80(8), 973 - 982 (2002).
  • A. K. Bhattacharya, F. Stolz And R. R. Schmidt, Design and synthesis of aryl/hetarylmethyl phosphonate-UMP derivatives as potential glucosyltransferase inhibitors, Tetrahedron Lett., 42, 5393 - 5395 (2001).
  • A. K. Bhattacharya And R. P. Sharma, Recent developments on the chemistry and biological activity of artemisinin and related antimalarials- an update, Heterocycles., 51, 1681 - 1745 (1999).
  • A. K. Bhattacharya, D. C. Jain And R. P. Sharma, Selective reduction of the exomethylene group of ?-methylene ?- or ?-lactones with CdCl2-Mg-MeOH-H2O, J. Chem. Res. (S)., , 768 - 769 (1998).
  • A. K. Bhattacharya, D. C. Jain, R. P. Sharma, R. Roy And A. T. McPhail, Boron trifluoride-acetic anhydride catalysed rearrangement of dihydroarteannuin B, Tetrahedron., 53(44), 14975 - 14990 (1997).