Publications

Research Group Publications

 
 
  • Vaibhav Ramachandra Pansare And Nagaraju Barsu*, Base-mediated denitrative C3-alkylation of quinoxaline deriv-atives, Organic and Biomolecular Chemistry., , (2024), DOI:https://doi.org/10.1039/D4OB01571A.
  • Nageswararao Moyilla, Ganeshdev Padhi And Deepti Kalsi* and Nagaraju Barsu* , Copper/Iron Co-Catalyzed Depolymerization of Post-Consumer Polycarbonate: A One-Pot Strategy to Synthesize Aryl Ethers, ACS Sustainable Chemistry & Engineering., , (2024), DOI:Just accepted.
  • Kishor V. Khopade, Nikhita S. Rajput, Raghavendrakumar Rangappa And Nagaraju Barsu * and Samir H. Chikkali *, Depolymerization of waste polyethylene to linear alkenes via sequential dehydrogenation and metathesis, Green Chemistry., 26, 10558 - 10566 (2024), DOI:https://doi.org/10.1039/D4GC03646H.
  • Ganeshdev Padhi, Vaibhav Ramachandra Pansare, Priyam Bajpai, Gamidi Rama Krishna, Kumar Vanka And and Nagaraju Barsu*, Depolymerization of Waste Polycarbonates to Value-Added Products, ChemSusChem., , e2024007 (2024), DOI:https://doi.org/10.1002/cssc.202400756.
  • M. Vijaykumar, C. Pradhan, R. G. Gonnade And B. Punji, Chelation-assisted and steric-controlled selectivity in the Pd-catalyzed C?H/C?H oxidative coupling of indoles, Chem. Commun., XX, XXXXX - XXXXX (2024), DOI:D4CC03835E.
  • M. Vijaykumar, R. G. Gonnade And B. Punji, Palladium-Catalyzed Regioselective C(4)?H Fluoroalkoxylation of Indoles through Weak Chelation Assistance, ChemCatChem., XX, XXXXX - XXXXX (2024), DOI:10.1002/cctc.202401188.
  • Manish Kumar And Pawan Kumar and Utpal Das*, Photocatalytic Oxidation of ?-Substituted Amines to Lactams/Amides, Advanced Synthesis & Catalysis., -, - - - (2024), DOI:10.1002/adsc.202400871.
  • Someshwar B. Kale, Tejaswini A patil And Utpal Das*, Rongalite as a C1 Source: Sulfonylmethylation of Indoles with Aryl/Alkyl- Hydrazides and Sulfinates, J. Org. Chem., 89, 11347 - 11352 (2024), DOI:10.1021/acs.joc.4c01012.
  • Archana Rai And Utpal Das*, Accessing meta-Enone-Substituted Anisoles using ArN2BF4 as Precatalyst via Rearrangement of Alkyne-Tethered Cyclohexadienones, Synthesis., 56, A - H (2024), DOI:10.1055/a-2331-9439.
  • Bagad, P. K.; Darole, R. S.; Krishna, G. R.; Senthilkumar And B, Highly Selective C-N and C-S Dual Functionalization of 1,3-Dicarbonyl Derivatives using TBHP as an Oxidant, J. Org. Chem., (Accepted), (2024), DOI:10.1021/acs.joc.4c00612.
  • Manisha Aher, Vaijayanti A. Kumar And Moneesha Fernandes , Implications of Natural 3'-5'- Linkages in the Loop Region of Isomeric 2'-5'-Linked Thrombin-Binding Aptamer, ChemistrySelect., 9, e202304254 (2024), DOI:10.1002/slct.202304254.
  • A. B. Shabade, R. K. Singh, R. G. Gonnade And B. Punji, Manganese-Catalyzed Chemoselective Direct Hydrogenation of ?,?-Epoxy Ketones and ?-Ketoamides at Room Temperature, Adv. Synth. Catal., XX, XXXXX - XXXXX (2024), DOI:10.1002/adsc.202400267.
  • S. M. Suryawanshi, S. Sahoo, P. S. Shaligram, N. Manna And R. C. Samanta*, Electrochemically enabled (3+2) cycloaddition of unbiased alkenes and ?-dicarbonyls, Chem. Commun., 60, 5836 - 5839 (2024), DOI:10.1039/d4cc01263a.
  • Kishor L. Handore, Heyuan Lu, Hyeongbin Park, Qingyu Xiong And and Robert A. Batey, Synthesis of N-Hydroxysuccinimide Esters, N-Acylsaccharins, and Activated Esters from Carboxylic Acids Using I2/PPh3, J. Org. Chem., , (2024), DOI:https://doi.org/10.1021/acs.joc.4c00272.
  • Shinde DR, Krishna GR And and Marelli UK, Metal-Free One-Pot Domino Synthesis of Oxazolidinethione Derivatives of Quaternary Amino Acids from ?-Amino Esters and Aldehydes Using CS2, J. Org. Chem., , (2024), DOI:https://doi.org/10.1021/acs.joc.3c02217.
  • Sunil L. Khamkar, Kishor L. Handore*, Harish M. Shinde And and D. Srinivasa Reddy*, Highly Stereoselective Diels–Alder-Based Strategy for the Synthesis of 3-epi-Formicin A and 1-epi-Formicin B, Organic Letters., ASAP, (2024), DOI:https://doi.org/10.1021/acs.orglett.4c01209.
  • S. B. Ankade, C. Pradhan, P. P. Samal, R. G. Gonnade, S. Krishnamurty And B. Punji, Iron-Catalyzed C–C and C–N Bond-Forming Tandem Amidation Offering Access to 3-Amino-3-Aminomethyl-2-Oxindole Frameworks, Adv. Synth. Catal., xxx, xxxx - xxxx (2024), DOI:10.1002/adsc.202400216.
  • C. Pradhan And B. Punji, Advancement in C–H Bond Alkylation of (Hetero)arenes Catalyzed by the Most Abundant Transition Metal - Iron, Org. Chem. Front., 11, 2397 - 2417 (2024), DOI:10.1039/D4QO00063C.
  • C. Pradhan And B. Punji, Book Chapter: Topics in Heterocyclic Chemistry on "Functionalisation of Heterocycles/Heteroaromatics through Transition Metal Catalysed C-H Activation" Chapter: Fe-Catalyzed Functionalization of Heterocycles through C-H Activation, Book Chapter, Springer., , (2024).
  • S. B. Ankade, S. Banerjee And B. Punji, Nickel-Catalyzed Branch Selective C-H Alkylation of Indoles and Azoles with Alkenes: An Additive- and Solvent-Free Approach, Eur. J. Org. Chem., xx, xxxx - xxxx (2024), DOI:10.1002/ejoc.202400376.
  • R. B. Pawar, M. H. Karmur And B. Punji, Ligand-free MnBr2-Catalyzed Chemo- and Stereoselective Hydroboration of Terminal Alkynes, Chem. Asian J., xx, xxxx - xxxx (2024), DOI:10.1002/asia.202400158.
  • S. Bansal And B. Punji, Chemodivergent Dehydrogenative Coupling of Alcohols by 3d Metal Catalysts, ChemCatChem., xx, xxxx - xxxx (2024), DOI:10.1002/cctc.202301558.
  • Darole, R. S.; Choudhary, S. S.; Sharma, H.; Mali, B. P.; Gopu, B.; Vanka, K.; Senthilkumar And B, Brønsted acid and Ni(II)-catalyzed C–H oxidation/ rearrangement of cyclotriveratrylenes (CTVs) to cyclic and acyclic quinones as potential anticancer agents, Org. Biomol. Chem., 22, 1038 - 1046 (2024), DOI:10.1039/d3ob01428b.
  • S. K. Verma And B. Punji, Copper-catalyzed regioselective C-H alkylation of phenol derivatives with unactivated alkyl chlorides: manifesting a Cu(I)/Cu(III) pathway, J. Catal., xx, xxxx - xxxx (2024), DOI:YJCAT_115351.
  • S. Bansal And B. Punji, Nickel-Catalyzed Chemodivergent Coupling of Alcohols: Efficient Routes to Access ?,?-Disubstituted Ketones and ?-Substituted Chalcones, Chem. Eur. J., xx, e202304082 (2024), DOI:rg/10.1002/chem.202304082.
  • Someshwar B. Kale, Manish Kumar, Dinesh R. Shinde, Gamidi Rama Krishna And Utpal Das*, Synthesis of N-functionalized 2,3-disubstituted benzofurans/naphthofurans from para-quinone methides and isocyanides via the [4 + 1] annulation pathway, Org. Chem. Front., 10, 3746 - 3751 (2023), DOI:10.1039/D3QO00048F.
  • Pawan Kumar, Archana Rai, Manish Kumar, Gamidi Rama Krishna And Utpal Das*, Radical Cascade Cyclization of Unactivated Alkene-Tethered Indoles with Aryldiazonium Salt and Sodium Metabisulfite to Access Azo- and Sulfonylated-2,3-Dihyro-1H-pyrrolo[1,2-a]indoles, J. Org. Chem., 13, 9123 - 9129 (2023), DOI:10.1021/acs.joc.3c00759.
  • Atish A. Wagh, Vaijayanti A. Kumar, Sapna Ravindranathan And Moneesha Fernandes, Unlike RNA-TBA (rTBA), iso-rTBA, the 2'–5'-linked RNA-thrombin-binding aptamer, is a functional equivalent of TBA, Chem. Commun., 59, 1461 - 1464 (2023), DOI:10.1039/d2cc05718b.
  • Darole, R. S.; Bagad, P. K.; Gonnade, R. G.; Alagarasu, K.; Punekar, M.; Shukla, S.; Parashar, D.; Senthilkumar And B, Synthesis of novel rhodamine type Anthrone Spiro-lactam (ASL) analogues and evaluation of antiviral activity against dengue and chikungunya viruses, Eur. J. Med. Chem., 261, 115849 (2023), DOI:https://doi.org/10.1016/ j.ejmech.2023.115849.
  • C. Pradhan, R. A. Jagtap, P. P. Samal, S. Krishnamurty And B. Punji, Iron-Catalyzed Regioselective C-H Alkylation of Indoles: An Additive-free Approach in Renewable Solvent, Green Chem., 25, 9733 - 9743 (2023), DOI:10.1039/D3GC03709F.
  • D. M. Sharma, A. B. Shabade, R. G. Gonnade And B. Punji, Manganese(I)-Catalyzed Chemoselective Transfer Hydrogenation of the C=C Bond in Conjugated Ketones at Room Temperature, Chem. Eur. J., 29, e202301174 (2023), DOI:10.1002/chem.202301174.
  • Devidas A. More, Sachin R. Shirsath And and M. Muthukrishnan, Metal- and Photocatalyst-Free, Visible-Light-Initiated C3 ?-Aminomethylation of Quinoxalin-2(1H)-ones via Electron Donor–Acceptor Complexes, The Journal of Organic Chemistry., 88, 133339 - 13350 (2023), DOI:https://doi.org/10.1021/acs.joc.3c01249.
  • Devidas A. More, Ganesh S. Ghotekar And Prof.?Dr. M. Muthukrishnan, BF3?Et2O-Catalyzed Selective C-4 Alkylation of Isoquinolin-1(2H)-ones Employing p-Quinone Methides, Chemistry–An Asian Journal., e202300546, (2023), DOI:https://doi.org/10.1002/asia.202200642.
  • Heyuan Lu, Kishor L. Handore, Tabitha Wood And Aaron D. Schimmer and Robert A. Batey, Total Synthesis of the 2,5-Disubstituted ?-Pyrone E1 UAE Inhibitor Himeic Acid A, Org. Lett., , (2023).
  • Priyanka Halder And Santosh B. Mhaske*, PIDA-mediated N–N bond formation to access pyrazolidine-3,5-diones: a novel process for uricosuric agents G-25671 and sulfinpyrazone, Chemical Communications., 59, 8242 - 8245 (2023), DOI:https://doi.org/10.1039/D3CC02078A.
  • Sameer R. Sonavane And Dr. Santosh B. Mhaske, Enantioselective Intramolecular Decarboxylative C?H Bond Func-tionalization of Quinazolinones with Amino Acids by Visible Light Photoredox Catalysis, Chemistry An Asian Journal., 18, (2023), DOI:https://doi.org/10.1002/asia.202300235.
  • Dangi A, Pande B, Agrawal S, Sarkar D, Vamkudoth KR And Marelli UK, Total synthesis, structure elucidation and expanded bioactivity of icosalide A: effect of lipophilicity and ester to amide substitution on its bioactivity, Org. Biomol. Chem., 21, 5725 - 5731 (2023), DOI:DOI https://doi.org/10.1039/D3OB00809F.
  • Dangi A And Marelli UK, Exploration of N?arylation of backbone amides as a novel tool for conformational modification in peptides, Chem. Eur. J., 29, (2023), DOI:https://doi.org/10.1002/chem.202301803.
  • I. Maksso, † R. C. Samanta, † Y. Zhan, K. Zhang, S. Warratz And L. Ackermann*, Polymer up-cycling by mangana-electrocatalytic C(sp3)–H azidation without directing groups, Chem. Sci., 14, 8109 - 8118 (2023), DOI:10.1039/D3SC02549G († contributed equally).
  • S. Bansal, R. G. Gonnade And B. Punji, Chemodivergent coupling of azoarenes with benzyl alcohols via borrowing hydrogen strategy using a well-defined nickel catalyst, Catal. Sci. Technol., 13, 2705 - 2713 (2023), DOI:10.1039/d3cy00090g.
  • Kishor V Khopade, Samir H Chikkali And Nagaraju Barsu, Metal-catalyzed plastic depolymerization, Cell Reports Physical Science., 4, 101341 (2023), DOI:doi.org/ 10.1016/j.xcrp.2023.101341.
  • M. Vijaykumar, C. Pradhan, R. G. Gonnade And B. Punji, Palladium-Catalyzed Chemoselective Oxygenation of C(sp2)-H and C(sp3)-H Bonds in Isatins, Org. Lett., 25, 1862 - 1867 (2023), DOI:10.1021/acs.orglett.3c00342.
  • C. Pradhan And B. Punji, Advances in the Iron-Catalyzed Direct Functionalizations of Heterocycles, Synlett., 34, 683 - 697 (2023), DOI:10.1055/a-1890-8503.
  • Siddharth K. Deepake, Manish Kumar, Pawan Kumar And Utpal Das*, alpha-Angelica Lactone Catalysed Oxidation of Pyrrolidines to Lactams, Eur. J. Org. Chem., , xxxx - xxxx (2022), DOI:10.1002/ejoc.202200712.
  • Mali, N.; Senthilkumar And B, Synthesis of Novel Biological Active 1,2,4,-Triazole Analogues, Chem. Proc., 4, 1 - 4 (2022), DOI:https://doi.org/10.3390/xxxxx.
  • 2. Mule, R.D.; Roy, R.; Mandal, K.; Chopra, D.; Dutta, T.; Sancheti, P.S.; Shinde, S.P.; Banerjee, S.; Koner, A.L.; Bhowal, R.; Senthilkumar, B.; Patil And N.T. , Interplay of Anion ??+ and ?+ ??+ Interactions in Novel Pyrido[2,1- Fluorescence Modulation and Applications in Live Cell Mitochondrial Imaging, Chem. Eur. J., , e202200632 (2022).
  • Mule, R. D.; Kumar, A.; Sancheti, S. P.; Senthilkumar, B.; Kumar, H.; Patil And N. T, BQ-AurIPr: a redox-active anticancer Au(I) complex that induces immunogenic cell death, Chem. Sci., 13, 10779 - 10785 (2022), DOI:DOI: 10.1039/d2sc03756d.
  • Vinita Yadav , Sayali G. Jagtap, Ekambaram Balaraman* And Santosh B. Mhaske*, Nickel-Catalyzed Direct Synthesis of N-Substituted Indoles from Amino Alcohols and Alcohols, Organic Letters., 24, 9054 - 9059 (2022), DOI:https://doi.org/10.1021/acs.orglett.2c03617.
  • Someshwar B. Kale, Popat K. Jori And Utpal Das*, Rongalite as a Sulfone Source: Sulfonylation of para -Quinone Methides and Alkyl/allyl Halides, Chemistry-An Asian Journal., xx, xxxx - xxxx (2022), DOI:10.1002/asia.202200408.
  • Kanungo SS, Mishra AK, Mhamane NB, Marelli UK, Kumar D And Gopinath CS, Possible Fine-Tuning of Methane Activation toward C2 Oxygenates by 3d-Transition Metal-Ions Doped Nano-Ceria-Zirconia, Inorg Chem., 61, 19577 - 19587 (2022), DOI:https://doi.org/10.1021/acs.inorgchem.2c03493.
  • Devidas A. More, M. Mujahid, M And Muthukrishnan*, Metal- And Light-Free Direct C-3 Ketoalkylation of Quinoxalin-2(1H)-Ones with Cyclopropanols in Aqueous Medium, ChemistrySelect., 7, e202203597 (2022), DOI:https://doi.org/10.1002/slct.202203597.
  • Sachin R. Shirsath, Devidas A. More And M. Muthukrishnan*, Metal-Free Aminocarbonylation of p-Quinone Methides with Isocyanides: Synthesis of Sterically Hindered ?-Arylated Acetamides, Chemistry—An Asian Journal., 17, e202200642 (2022), DOI:https://doi.org/10.1002/asia.202200642.
  • A. B. Shabade, D. M. Sharma, P. Bajpai, R. G. Gonnade, K. Vanka And B. Punji, Room Temperature Chemoselective Hydrogenation of C=C, C=O and C=N Bonds by Using a Well-Defined Mixed Donor Mn(I) Pincer Catalyst, Chem. Sci., 13, 13764 - 13773 (2022), DOI:10.1039/D2SC05274A.
  • D. M. Sharma, C. Gouda, R. G. Gonnade And B. Punji, Room Temperature Z-selective Hydrogenation of Alkynes by Hemilabile and Non-innocent (NNN)Co(II) Catalyst, Catal. Sci. Technol., 12, 1843 - 1849 (2022), DOI:10.1039/D2CY00027J.
  • R. A. Jagtap, C. Pradhan, R. G. Gonnade And B. Punji, An Efficient Route to 3,3'-Biindolinylidene-diones by Iron-Catalyzed Dimerization of Isatins, Chem. Asian J., 17, xxxx - xxxx (2022), DOI:10.1002/asia.202200414.
  • S. K. Verma And B. Punji, Manganese-Catalyzed C(sp2)-H Alkylation of Indolines and Arenes with Unactivated Alkyl Bromides, Chem. Asian J., 17, e202200103 (2022), DOI:10.1002/asia.202200103.
  • S. Sudhakaran, P. G. Shinde, E. K. Aratikatla, S. H. Kaulage, P. Rana, R. S. Parit, D. S. Kavale, B. Senthilkumar And B. Punji, Nickel-Catalyzed Asymmetric Hydrogenation for the Synthesis of Key Sitagliptin Intermediate, Chem. Asian J., 17, e202101208 (2022), DOI:10.1002/asia.202101208.
  • Lakshmi Goswami‡, Lovely Gupta‡, Sayantan Paul, Maansi Vermani And Pooja Vijayaraghavan* and Asish K. Bhattacharya*, Design and synthesis of eugenol/isoeugenol glycoconjugates and other analogues as antifungal agents against Aspergillus fumigatus†, RSC Med. Chem., , (2022), DOI:DOI: 10.1039/D2MD00138A.
  • Lovely Gupta, Pooja Sen, Asish K. Bhattacharya And Pooja Vijayaraghavan, Isoeugenol affects expression pattern of conidial hydrophobin gene RodA and transcriptional regulators MedA and SomA responsible for adherence and biofilm formation in Aspergillus fumigatus, Archives of Microbiology (Springer)., 204:214, 1 - 14 (2022), DOI:https://doi.org/10.1007/s00203-022-02817-w.
  • R. Mei, R. C. Samanta, U. Dhawa, W. Ma And L. Ackermann, Electrochemical Cobalt-Catalyzed C–H Activations with Potential, in The Chemistry of Organocobalt Chemistry (Eds.: C. Gosmini, I. Marek), Wiley-VCH, Weinheim., , (2022).
  • Suhag S. Patil, Gorakhnath R. Jachak, Gamidi Rama Krishna, Narshinha P. Argade And * D. Srinivasa Reddy*, Total Synthesis of 12,13-Dibenzyl-Banistenoside B and Analogs, Eur J Org Chem., 2022, e202200222 (2022), DOI:doi.org/10.1002/ejoc.202200222.
  • Rahul D. Shingare, John B. MacMillan And D. Srinivasa Reddy* , Antibiotic natural product hunanamycin A: Lead identification towards anti-Salmonella agents, Eur J Med Chem., 236, 114245 (2022), DOI:10.1016/j.ejmech.2022.114245.
  • Yash Mankad, Sagar S. Thorat, Pronay Das, Gamidi Rama Krishna, Ravindar Kontham And * D. Srinivasa Reddy* , Ready Access to Benzannulated [5,5]-Oxaspirolactones Using Au(III)-Catalyzed Cascade Cyclizations, J. Org. Chem., 87, 3025 - 3041 (2022), DOI:doi.org/10.1021/acs.joc.1c02843.
  • Kritee Mehdiratta, Shubham Singh, Sachin Sharma, Rashmi S. Bhosale, Rahul Choudhury, Dattatraya P. Masal, Alzu Manocha, Bhushan Dilip Dhamale, Naseem Khan, Vivekanand Asokachandran, Pooja Sharma, Melanie Ikeh, Amanda C. Brown, Tanya Parish, Anil K. Ojha, Joy Sarojini Michael, Mohammed Faruq, Guruprasad R. Medigeshi, Debasisa Mohanty, D. Srinivasa Reddy, Vivek T. Natarajan, Siddhesh S. Kamat And Rajesh S. Gokhale, Kupyaphores are zinc homeostatic metallophores required for colonization of Mycobacterium tuberculosis, PNAS., 119, e211029311 (2022), DOI:doi.org/10.1073/pnas.2110293119.
  • Mule, R.D.; Kumar, A.; Sancheti, P.S.; Senthilkumar, B.; Ku-mar, H.; Patil And N.T, BQ-AurIPr: A Redox-Active Anticancer Au(I) Complex that Induces Immunogenic Cell Death in Non-Small Cell Lung Cancer, ChemRxiv., , (2022), DOI:10.26434/chemrxiv-2022-m3xxx.
  • Sudhakaran, S.; Shinde, G.P.; Aratikatla, K.E.; Kaulage, H.S.; Rana, P.; Parit, R.S.; Kavale, S.D.; Senthilkumar, B.; Punji And B, Nickel-Catalyzed Asymmetric Hydrogenation for the Synthesis of a Key Intermediate of Sitagliptin, Chem Asian J., 17, e2021012 (2022), DOI:10.1002/asia.202101208.
  • Dattatraya P. Masal, Rahul Choudhury, Aman Singh And D. Srinivasa Reddy*, Ready Access to Densely Substituted Furans Using Tsuji?WackerType Cyclization, J. Org. Chem., 87, 556 - 558 (2022), DOI:doi.org/10.1021/acs.joc.1c02567.
  • Wagh A. A, Ghalawat M. And Fernandes M, Replacement of Loop Residues in TBA by an Abasic Ethylene Glycol Spacer: Effect on Stability, Structure and Function, ChemistrySelect., 6, 10648 - 10650 (2021), DOI:https://doi.org/10.1002/slct.202102269.
  • S. Ghosh, K. B. Cotta, A. A. Hande, M. Fernandes And S. Mehra, PNA-mediated efflux inhibition as a therapeutic strategy towards overcoming drug resistance in Mycobacterium smegmatis, Microbial Pathogenesis., 151, 104737 (2021).
  • Alam MN, Dash SR, Mukherjee A, Pandole S, Marelli UK, Vanka K And Maity P, [1,3]-Claisen Rearrangement via Removable Functional Group Mediated Radical Stabilization, Org Lett., 23, 890 - 895 (2021), DOI:https://doi.org/10.1021/acs.orglett.0c04109.
  • Sachin R. Shirsath, Sagar M. Chandgude And M. Muthukrishnan*, Iron catalyzed tandem ring opening/1,6-conjugate addition of cyclopropanols with p-quinone methides: new access to ?,?-diaryl ketones, Chemical Communications., 57, 13582 - 13585 (2021), DOI:https://doi.org/10.1039/D1CC05997A.
  • T. H. Meyer, † R. C. Samanta, † A. Del Vecchio And L. Ackermann* , Mangana(III/IV)electro-Catalyzed C(sp3)–H Azidation, Chem. Sci., 12, 2890 - 2897 (2021), DOI:10.1039/d0sc05924b († contributed equally).
  • Eswar K. Aratikatla, Md Kalamuddin, Kalpeshkumar C. Rana, Gaurav Datta, Mohd Asad, Srividhya Sundararaman, Pawan Malhotra, Asif Mohmmed And Asish K. Bhattacharya, Combating multi-drug resistant malaria parasite by inhibiting falcipain-2 and heme-polymerization: Artemisinin-peptidyl vinyl phosphonate hybrid molecules as new antimalarials, European Journal of Medicinal Chemistry., 220, (2021), DOI:https://doi.org/10.1016/j.ejmech.2021.113454.
  • Rajib Mandal, Nagaraju Barsu, Bholanath Garai, Abir Das And Dmitry Perekalin and Basker Sundararaj, Room Temperature C-H Bond Alkynylation by Merging Cobalt and Photo-redox catalysis, Chem. Commun., 57, 12167 - 12170 (2021), DOI:DOI https://doi.org/10.1039/D1CC05263B.
  • R. C. Samanta And L. Ackermann* , Evolution of Earth-Abundant 3d-Metallaelectro-Catalyzed C–H Activation: From Chelation-Assistance to C–H Functionalization without Directing Groups, Chem. Rec., 21, 2430 - 2441 (2021), DOI:10.1002/tcr.202100096.
  • K. Korvorapun, R. C. Samanta, T. Rogge And L. Ackermann* , Remote C–H Functionalizations by Ruthenium Catalysis, Synthesis., 53, 2911 - 2946 (2021), DOI:10.1055/a-1485-5156.
  • K. Korvorapun, R. C. Samanta, T. Rogge And L. Ackermann, Ruthenium-Catalyzed Remote C–H Functionalizations, in Remote C–H bond Functionalizations (Eds.: D. Maiti, S. Guin), Wiley-VCH, Weinheim., , (2021).
  • AkshayS.Kulkarni, RemyaRamesh, SafalWalia, ShahebazI.Sayyad, GaneshB.Gathalkar, SeetharamsingBalamkundu, ManaliJoshi, AvalokiteswarSen And *andD.SrinivasaReddy*, Identification of a Novel Series of Potent Organosilicon Mosquito Repellents, ACSOmega., 6, 31236 - 31243 (2021), DOI:doi.org/10.1021/acsomega.1c04961.
  • Akshay S. Kulkarni, Remya Ramesh, Safal Walia, Shahebaz I. Sayyad, Ganesh B. Gathalkar, Seetharamsing Balamkundu, Manali Joshi, Avalokiteswar Sen And and D. Srinivasa Reddy, Identification of a Novel Series of Potent Organosilicon Mosquito Repellents, ACS OMEGA., 6(46), 31236 - 31243 (2021), DOI:https://doi.org/10.1021/acsomega.1c04961.
  • S. B. Ankade, P. P. Samal, V. Soni, R. G. Gonnade, S. Krishnamurty And B. Punji, Ni(II)-Catalyzed Intramolecular C–H/C–H Oxidative Coupling: An Efficient Route to Functionalized Cycloindolones and Indenoindolones, ACS Catal., 11, 12384 - 12393 (2021), DOI:10.1021/acscatal.1c03314.
    Highlighted in "Synfacts, 2021, 17, 1357" by Prof. Mark Lautens
  • Aboli Girme*, Ganesh Saste, Sandeep Pawar, Chetana Ghule, Amit Mirgal, Saurabh Patel, Anshuly Tiwari, Sautik Ghoshal, Sandip B. Bharate, Sonali S. Bharate, D. Srinivasa Reddy, Ram A. Vishwakarma And and Lal Hingorani, Quantitative Determination and Characterization of a Kashmir Saffron (Crocus sativus L.)-Based Botanical Supplement Using Single-Laboratory Validation Study by HPLC-PDA with LC–MS/MS and HPTLC Investigations, ACS Omega., 6, 23460 - 23474 (2021), DOI:doi.org/10.1021/acsomega.1c03470.
  • Rama Krishna Gamidi, Monica Dandawate, Srinu Tothadi, Rahul Choudhury, Ashwini K. Nangia And D. Srinivasa Reddy, Separation of a diastereomeric diol pair using the mechanical properties of crystals, CrystEngComm., 23, 7056 - 7060 (2021), DOI:doi.org/10.1039/D1CE01055G.
  • Bhagavatula L. V. Prasad, Prathap C. Sivasankaran, Pitamber Patel, Pushpa V. Malekar, K. V. Maya And Chepuri V. Ramana, Synthesis of anisotropic rod-like gold nanostructures in organic media, J. Chem. Sci., 133, - - - (2021), DOI:org/10.1007/s12039-021-01952-z.
  • Sibadatta Senapati, Shyamsundar Das, Ruchi Dixit, Kumar Vanka And Chepuri V. Ramana*, Synthesis of four diastereomers of notoryne and their 13C NMR chemical shifts analysis, J. Chem. Sci., 133, - - - (2021), DOI:org/10.1007/s12039-021-01929-y.
  • Pawan S. Dhote, Kishor Pund And Chepuri V. Ramana*, Intermolecular Interception of ?-Oxo Gold Carbenes of Nitroalkyne Cycloisomerization with 1,2-Benzo[d]isoxazole: Synthesis of Functionalized Quinazoline 1-Oxides, J. Org. Chem., 86, 10874 - 10882 (2021), DOI:org/10.1021/acs.joc.1c01221.
  • Pawan S. Dhote, Swapnil V. Halnor And Chepuri V. Ramana*, Gold?Catalysed Nitroalkyne Cycloisomerization–Synthetic Utility, Chem. Rec., -, - - - (2021), DOI:org/10.1002/tcr.202100111.
  • Sibadatta Senapati, Nivedya A. Unmesh, Manoj Shet, Iram Ahmad, Nandu Ajikumar And Chepuri V. Ramana*, Unified Approach for the Total Synthesis of Bis-THF C15 Acetogenins: A Chloroenyne from Laurencia majuscula, Laurendecumenyne B and Laurefurenynes A/B, Synthesis., 53, 2903 - 2910 (2021), DOI:10.1055/a-1500-1407.
  • Pawan S. Dhote And Chepuri V. Ramana*, Interrupting the [Au]-Catalyzed Nitroalkyne Cycloisomerization: Trapping the Putative ?-Oxo Gold Carbene with Benzo[c]isoxazole, Org. Lett., 23, 2632 - 2637 (2021), DOI:org/10.1021/acs.orglett.1c00539.
  • Pawan S. Dhote, Pitamber Patel, Kumar Vanka And Chepuri V. Ramana*, Total synthesis of the pseudoindoxyl class of natural products, Org. Biomol. Chem., 19, 7970 - 7994 (2021), DOI:org/10.1039/D1OB01285A.
  • Vipin K. Raj, Pawan S. Dhote, Kumar Vanka And Chepuri V. Ramana*, Gold-Catalyzed Complementary Nitroalkyne Internal Redox Process: A DFT Study, Front. Chem., 9, 689780 (2021), DOI:org/10.3389/fchem.2021.689780.
  • Ganesh V. More, Pushpa V. Malekar, Rupali G. Kalshetti, Mahesh H. Shinde And Chepuri V. Ramana*, Ru-Catalyzed Asymmetric Transfer Hydrogenation of ?-Acyl Butyrolactone via Dynamic Kinetic Resolution: Asymmetric Synthesis of bis-THF Alcohol Intermediate of Darunavir, Tetrahedron Lett., 66, 152831 - 152835 (2021), DOI:org/10.1016/j.tetlet.2021.152831.
  • Sibadatta Senapati And Chepuri V. Ramana*, A concise/catalytic approach for the construction of the C14–C28 fragment of eribulin, Org. Biomol. Chem., 19, 4542 - 4550 (2021), DOI:org/10.1039/D1OB00661D.
  • Paresh R. Athawale, Vishal Zade, Gamidi Rama Krishna And D. Srinivasa Reddy*, Tuning of ?-Silyl Carbocation Reactivity into Enone Transposition: Application to the Synthesis of Peribysin D, E-Volkendousin, and E-Guggulsterone, Org. Lett., 23, 6642 - 6647 (2021), DOI:10.1021/acs.orglett.1c02173.
  • M. Vijaykumar And B. Punji, Pd(II)-Catalyzed Chemoselective Acetoxylation of C(sp2)-H and C(sp3)-H Bonds in Tertiary Amides, J. Org. Chem., 86, 8172 - 8181 (2021), DOI:10.1021/acs.joc.1c00629.
  • T. Rogge, N. Kaplaneris, N. Chatani, J. Kim, S. Chang, B. Punji, L. L. Schafer, D. G. Musaev, J. Wencel-Delord, C. A. Roberts, R. Sarpong, Z. E. Wilson, M. A. Brimble, M. J. Johansson And L. Ackermann, C-H Activation, Nature Rev. Meth. Primers., 1, 43 (2021), DOI:10.1038/s43586-021-00041-2.
  • S. B. Ankade, A. B. Shabade, V. Soni And B. Punji, Unactivated Alkyl Halides in Transition-Metal-Catalyzed C-H Bond Alkylation, ACS Catal., 11, 3268 - 3292 (2021), DOI:10.1021/acscatal.0c05580.
  • M. Vijaykumar And B. Punji, Advances in Transition-Metal-Catalyzed C–H Bond Oxygenation of Amides, Synthesis., 53, 2935 - 2946 (2021), DOI:10.1055/a-1481-2584.
  • R. A. Jagtap, S. B. Ankade, R. G. Gonnade And B. Punji, Achiral and Chiral NNN-Pincer Nickel Complexes with Oxazolinyl Backbone: Application in Transfer Hydrogenation of Ketones, New J. Chem., 45, 11927 - 11936 (2021), DOI:10.1039/D1NJ01698A.
  • D. M. Sharma And B. Punji, Nickel-Catalysed Benzylic C–H Functionalization, Book Chapter for "Handbook of CH-Functionalization (CHF)"., xx, xxxxx - xxxxx (2021), DOI:xxxxxxxxxxx.
  • Vinita Yadav, Ekambaram Balaraman And Santosh B. Mhaske, Phosphine-Free Manganese(II)-Catalyst Enables Acceptorless Dehydrogenative Coupling of Alcohols with Indoles, Advanced Synthesis & Catalysis., 363, (2021), DOI:https://doi.org/10.1002/adsc.202100621.
  • Amol B. Viveki, § Mahesh D. Pol, § Priyanka Halder, Sameer R. Sonavane And Santosh B. Mhaske*, Annulation of Enals with Carbamoylpropiolates via NHC-Catalyzed Enolate Pathway: Access to Functionalized Maleimides/Iso-maleimides and Synthesis of Aspergillus FH-X-213, J. Org. Chem., 86,14, 9466 - 9477 (2021), DOI:https://doi.org/10.1021/acs.joc.1c00782.
  • Pawan Kumar, Someshwar B. Kale, Rajesh G. Gonnade And Utpal Das*, Acid Mediated Sulfonylation of para-Quinone Methides with Tosylmethyl Isocyanides for the Synthesis of Diarylmethyl Sulfones, ChemistrySelect., 6, 7158 - 7161 (2021), DOI:10.1002/slct.202102272.
  • Paresh R. Athawale, Hanuman P. Kalmode And D. Srinivasa Reddy*, DBU/O2?Mediated Oxidation of Dienones, J. Org. Chem., 86, 9200 - 9205 (2021), DOI:10.1021/acs.joc.1c00529.
  • Rahul Choudhury And D. Srinivasa Reddy*, Total Synthesis of a Hypothetical Macroketone of Migrastatin, Eur. J. Org. Chem., 2021, 3050 - 3053 (2021), DOI:10.1002/ejoc.202100484.
  • Palak Babbar, Pronay Das, Yogavel Manickam, Yash Mankad, Swati Yadav, Suhel Parvez, Amit Sharma* And D Srinivasa Reddy* , Design, Synthesis, and Structural Analysis of Cladosporin-Based Inhibitors of Malaria Parasites, ACS Infect. Dis., 7, 1777 - 1794 (2021), DOI:10.1021/acsinfecdis.1c00092.
  • Pronay Das And D Srinivasa Reddy* , Total synthesis of twelve membered resorcyclic acid lactones,(R)-penicimenolide A, (R)-resorcyclide and (R)-dihydroresorcyclide, Tetrahedron., 85, 132059 (2021), DOI:10.1016/j.tet.2021.132059.
  • Akshay S. Kulkarni And Eagala Ramesh D. Srinivasa Reddy*, One?Pot Oxidation of Secondary Alcohols to ??Hydroxy Ketones: Application to Synthesis of Oxoaplysinopsin D, E, F, & G, Eur. J. Org. Chem., 15, 2188 - 2192 (2021), DOI:10.1002/ejoc.202100184.
  • Dr. Gorakhnath R. Jachak, Drishya Elizebath, Dr. Anurag Shukla, Dr. Dhanasekaran Shanmugam And * D Srinivasa Reddy*, Synthesis and Biological Evaluation of Hoshionolactam?Based Compounds, Eur. J. Org. Chem., 15, 2212 - 2218 (2021), DOI:10.1002/ejoc.202001588.
  • Ranjit S. Atapalkar, Paresh R. Athawale, D. Srinivasa Reddy* And Amol A. Kulkarni* , Scalable, sustainable and catalyst-free continuous flow ozonolysis of fatty acids, Green Chem., 23, 2391 - 2396 (2021), DOI:10.1039/D0GC04021E.
  • Yash Mankad, Pronay Das, Ejaj Pathan, MV Deshpande And D Srinivasa Reddy* , Herbicidal bio-assay of isocladosporin enantiomers and determination of its plausible absolute configuration, J Antibiot., 74, 280 - 284 (2021), DOI:10.1038/s41429-020-00391-1.
  • Ruyi Zhang, Lisanne Noordam, Xumin Ou, Buyun Ma, Yunlong Li, Pronay Das, Shaojun Shi, Jiaye Liu, Ling Wang, Pengfei Li, Monique MA Verstegen, D Srinivasa Reddy, Luc JW van Der Laan, Maikel P Peppelenbosch, Jaap Kwekkeboom, Ron Smits And Qiuwei Pan, The biological process of lysine?tRNA charging is therapeutically targetable in liver cancer, Liver Int., 41, 206 (2021), DOI:doi.org/10.1111/liv.14692.
  • Md Nirshad Alam, Soumya Ranjan Dash, Anirban Mukherjee, Satish Pandole, Udaya Kiran Marelli, Kumar Vanka And Pradip Maity*, [1,3]-Claisen Rearrangement via Removable Functional Group Mediated Radical Stabilization, Organic Letters., 23, 890 - 895 (2021), DOI:10.1021/acs.orglett.0c04109.
  • Soniya Rani, Soumya Ranjan Dash, Asish Bera, Md Nirshad Alam, Kumar Vanka And Pradip Maity, Phosphite mediated asymmetric N to C migration for the synthesis of chiral heterocycles from primary amines, Chemical Science., 12, 8996 - 9003 (2021), DOI:10.1039/D1SC01217G.
  • R. A. Jagtap And B. Punji, Nickel-Catalyzed C-H Bond Functionalization of Azoles and Indoles, Chem. Rec., xx, xxxx - xxxx (2021), DOI:10.1002/tcr.202100113.
  • S. Bansal, A. B. Shabade And B. Punji, Advances in C(sp2)–H/C(sp2)–H Oxidative Coupling of (Hetero)arenes using 3d Transition Metal Catalysts, Adv. Synth. Catal., 363, 1998 - 2022 (2021), DOI:10.1002/adsc.202001498.
  • M. N. Aher, N. D. Erande, V. A. Kumar, M. Fernandes And R. G. Gonnade, Influence of fluorine substitution on the molecular conformation of 3'-deoxy-3'-fluoro-5-methyluridine, Acta Crystallogr. C. Struct. Chem., 76, 346 - 352 (2020), DOI:https://doi.org/10.1107/S2053229620003083.
  • M. Varada, M. Aher, N. Erande, V. A. Kumar And M. Fernandes, Methoxymethyl Threofuranosyl Thymidine (4?-MOM-TNA-T) at the T7 Position of the Thrombin-Binding Aptamer Boosts Anticoagulation Activity, Thermal Stability, and Nuclease Resistance, ACS Omega., 5, 498 - 506 (2020).
  • Darole, R. S. Britto, C. D.; Mukherjee, A.; Gonnade, R. G.; Sekar, K.; Senthilkumar And B. , Anthrone-spirolactam and quinoline hybrid based sensor for selective detection of Fe3+ ions in water samples, Appl. Organomett. Chem., 34, e5867 (2020), DOI:10.1002/aoc.5867.
  • Aegurl, B.; Ram D. Mandle, R. D.; Shinde, P. G.; Parit, R. S.; Kamble, S. P.; Sudalai, A.; Senthilkumar And B. , Triethyl Phosphite/Benzoyl Peroxide Mediated Reductive Dealkylation of O-Benzoylhydroxylamines: A Cascade Synthesis of Secondary Amides, Eur. J. Org. Chem., , 4235 - 4238 (2020).
  • Andy A. Tjeng; Kishor L. Handore and Robert A. Batey, Stereocontrolled Microwave Assisted Domino [3,3]-Sigmatropic Reactions: A Winstein-Overman Rearrangement for the Formation of Differentiated Contiguous C–N Bonds, Org. Lett., 22, 3050 - 3055 (2020).
  • Dangi A, Balmik AA, Ghorpade AK, Gorantla NV, Sonawane SK, Chinnathambi S And Marelli UK, Residue-based propensity of aggregation in the Tau amyloidogenic hexapeptides AcPHF6* and AcPHF6, RSC Adv., 10, 27331 - 27335 (2020), DOI:DOI https://doi.org/10.1039/D0RA03809A.
  • Balmik AA, Chidambaram H, Dangi A, Marelli UK And Chinnathambi S, HDAC6 ZnF UBP as the Modifier of Tau Structure and Function, Biochemistry., 59, 4546 - 4562 (2020), DOI:https://doi.org/10.1021/acs.biochem.0c00585.
  • Balmik AA, Das R, Dangi A, Gorantla NV, Marelli UK And Chinnathambi S, Melatonin interacts with repeat domain of Tau to mediate disaggregation of paired helical filaments, Biochim Biophys Acta Gen Subj., 1864, 129467 (2020), DOI:https://doi.org/10.1016/j.bbagen.2019.129467.
  • Sonawane SK, Chidambaram H, Boral D, Gorantla NV, Balmik AA, Dangi A, Ramasamy S, Marelli UK And Chinnathambi S, EGCG impedes human Tau aggregation and interacts with Tau, EGCG impedes human Tau aggregation and interacts with Tau., 10, 12579 (2020), DOI:https://doi.org/10.1038/s41598-020-69429-6.
  • Dan VM, J S V, C J S, Sanawar R, Lekshmi A, Kumar RA, Santhosh Kumar TR, Marelli UK, Dastager SG And Pillai MR, Molecular Networking and Whole-Genome Analysis Aid Discovery of an Angucycline That Inactivates mTORC1/C2 and Induces Programmed Cell Death, ACS Chem Biol., 15, 780 - 788 (2020), DOI:https://doi.org/10.1021/acschembio.0c00026.
  • Meena CL, Singh D, Weinmüller M, Reichart F, Dangi A, Marelli UK, Zahler S And Sanjayan GJ, Novel cilengitide-based cyclic RGD peptides as ?v?3 integrin inhibitors, Bioorg Med Chem Lett., 30, 127039 (2020), DOI:https://doi.org/10.1016/j.bmcl.2020.127039.
  • Das TK, Madica K, Krishnan J, Marelli UK And Biju AT, Heterocyclic Carbene Catalysis Exploiting Oxidative Imine Umpolung for the Generation of Imidoyl Azoliums, J Org Chem., 85, 5114 - 5121 (2020), DOI:https://doi.org/10.1021/acs.joc.0c00360.
  • Sachin R. Shirsath, Ganesh S. Ghotekar, Vir Bahadur, Rajesh G. Gonnade And M. Muthukrishnan*, Silver-Catalyzed Cascade Cyclization/1,6-Conjugate Addition of Homopropargyl Sulfonamides to p-Quinone Methides: An Approach to Diverse 3-Diarylmethine Substituted Dihydropyrroles, The Journal of Organic Chemistry., 85, 15038 - 15050 (2020), DOI:https://doi.org/10.1021/acs.joc.0c01922.
  • Tharun K. Kotammagari, Sayantan Paul, Ganesh K. Barik And Manas K. Santra and Asish K. Bhattacharya, Synthesis of artemisinic acid derived glycoconjugates and their anticancer studies, Organic & Biomolecular Chemistry., , 1 - 13 (2020), DOI:DOI: 10.1039/D0OB00216J.
  • Eswar K. Aratikatla, Md Kalamuddin, Pawan Malhotra, Asif Mohmmed And * and Asish K. Bhattacharya*, Enantioselective Synthesis of ??Phenyl-?-amino Vinyl Phosphonates and Sulfones and Their Application to the Synthesis of Novel Highly Potent Antimalarials, ACS Omega., 5, 29025 - 29037 (2020), DOI:https://dx.doi.org/10.1021/acsomega.0c03470.
  • Nagaraju Barsu, Markus Leutzsch And and Alois Fürstner*, Ruthenium-Catalyzed trans-Hydroalkynylation and trans-Chloroalkynylation of Internal Alkynes, J. Am. Chem. Soc., 142, 18746 - 18752 (2020), DOI:https://doi.org/10.1021/jacs.0c08582.
  • R. Mei*, U. Dhawa, R. C. Samanta, W. Ma, J. Wencel-Delord* And L. Ackermann* , Cobalt–Catalyzed Oxidative C–H Activation: Strategies and Concepts, ChemSusChem., 13, 3306 - 3356 (2020), DOI:10.1002/cssc.202000024.
  • S.-K. Zhang, R. C. Samanta, A. Del Vecchio And L. Ackermann* , Evolution of High-Valent Nickelaelectro-Catalyzed C–H Activation: From Cross(-Electrophile)-Couplings to Electrooxidative C–H Transformations, Chem. Eur. J., 26, 10936 - 10947 (2020), DOI:10.1002/chem.202001318.
  • R. C. Samanta, T. H. Meyer, I. Siewert And L. Ackermann* , Renewable Resources for Sustainable Metallaelectro-Catalysed C–H Activation, Chem. Sci., 11, 8657 - 8670 (2020), DOI:10.1039/d0sc03578e.
  • R. C. Samanta, J. Struwe And L. Ackermann* , Nickelaelectro-Catalyzed Mild C–H Alkylations at Room Temperature, Angew. Chem. Int. Ed., 59, 14154 - 14159 (2020), DOI:10.1002/anie.202004958.
  • Banerjee, S.; Ambegave, S. B.; Mule, R. D.; Senthilkumar, B.; Patil And N. T, Gold-Catalyzed Alkynylative Meyer-Schuster Rearrangement, Org. Lett., 22(12), 4792 - 4796 (2020).
  • Mahesh H.Shinde And Chepuri V. Ramana*, An Apparent Umpolung Reactivity of Indole via [Au]?Catalysed Cyclisation and Lewis?Acid Mediated Allylation, Chem. Eur. J., 26, 17171 - 17175 (2020), DOI:10.1002/chem.202003441.
  • Ejaj K.Pathan, Anand M. Kulkarni, Prasanna V. L. Nallaballe, Chepuri V. Ramana And Mukund V. Deshpande, NADP-dependent glutamate dehydrogenases in a dimorphic zygomycete Benjaminiella poitrasii: Purification, characterization and their evaluation as an antifungal drug target, Biochim. Biophys. Acta., 1864, 129696 (2020), DOI:org/10.1016/j.bbagen.2020.129696.
  • Shaziya K. Siddiqui, Vinod J. SahayaSheela , Kolluru Srinivas, Ganesh N. Pandian, Thankayyan R. Santhoshkumar, Vipin M. Dan And Chepuri V. Ramana*, Discovery of 3-(benzofuran-2-ylmethyl)-1H-indole derivatives as potential autophagy inducers in cervical cancer cells, Bioorg. Med. Chem. Lett., 30, 127431 - 127435 (2020), DOI:org/10.1016/j.bmcl.2020.127431.
  • Venakannababu Mullapudi And Chepuri V. Ramana*, Attempted Synthesis of Central Furopyran Core of Diocolletines A via a Gold-Catalyzed Cascade 1, 6-Diyne Cycloisomerization Process, Tetrahedron Letters., 61, 152367 - 152370 (2020), DOI:org/10.1016/j.tetlet.2020.152367.
  • Venkannababu Mullapudi, Iram Ahmad, Sibadatta Senapati And Chepuri V. Ramana*, Total Synthesis of (+)-Petromyroxol, (?)-iso-Petromyroxol, and Possible Diastereomers, ACS Omega., 5, 25334 - 25348 (2020), DOI:org/10.1021/acsomega.0c03674.
  • Rupali G. Kalshetti And Chepuri V. Ramana*, Oxidative Rearrangement of Stilbenes to 2, 2-Diaryl-2-hydroxyacetaldehydes, ACS Omega., 5, 25199 - 25208 (2020), DOI:org/10.1021/acsomega.0c03328.
  • Monica Dandawate, Rahul Choudhury, Gamidi Rama Krishna And D. Srinivasa Reddy*, Total synthesis and absolute configuration determination of Ktedonoketone, a benzenoid metabolite from Thermophilic bacterium, Tetrahedron Letters., 61, 152526 (2020), DOI:10.1016/j.tetlet.2020.152526.
  • Chinnakuzhanthai Gangadurai, Giri Teja Illa And D. Srinivasa Reddy* , FeCl3-catalyzed oxidative decarboxylation of aryl/heteroaryl acetic acids: preparation of selected API impurities, Org. Biomol. Chem., 18, 8459 - 8466 (2020), DOI:10.1039/D0OB01790F.
  • Vidya B. Gunjal, Ritesh Thakare, Sidharth Chopra* And D. Srinivasa Reddy* , Teixobactin: A Paving Stone toward a New Class of Antibiotics, J. Med. Chem., 63, 12171 - 12195 (2020), DOI:10.1021/acs.jmedchem.0c00173.
  • Rajeshwari Tiwari, Prashant Suresh Shinde, Sreejesh Sreedharan, Anik Kumar Dey, Katherine Vallis, Santosh B. Mhaske, Sumit Kumar Pramanik And Amitava Das, "Photoactivable Prodrug for Simultaneous Release of Mertansine, and CO along with a BODIPY Derivative as a Luminescent Marker in Mitochondria: A Proof of Concept for NIR Image-Guided Cancer Therapy", Chemical Science., Just Accepted, (2020).
  • Priyanka Halder, Mahesh D. Pol, Milind M Ahire And Santosh B. Mhaske , "Construction of Unique SCF3-Containing Building Blocks via Allylic Alkylation of Morita-Baylis-Hillman Adducts", Org. Biomol. Chem., 18, 2085 - 2093 (2020).
  • Ganesh S. Ghotekar, Sachin R. Shirsath And Aslam C. Shaikh and M. Muthukrishnan*, 1,6-Conjugate addition initiated formal [4+2] annulation of p-quinone methides with sulfonyl allenols: a unique access to spiro[5.5]undeca-1,4-dien-3-one scaffolds, Chemical Communications., 56, 5022 - 5025 (2020), DOI:https://doi.org/10.1039/D0CC01005G.
  • Sravanya Konchada, Naresh Killi, Shahebaz Sayyad, Ganesh B. Gathalkar And Rathna V. N. Gundloori, Blends of neem oil based polyesteramide as nanofiber mats to control Culicidae, RSC Advances., 10 (70), 42827 - 42837 (2020), DOI:https://doi.org/10.1039/D0RA08297J.
  • Thanusha Thatikonda, ‡ Siddharth K. Deepake‡ Pawan Kumar And Utpal Das*, alpha-Angelica lactone catalyzed oxidation of benzylic sp3 C–H bonds of isochromans and phthalans, Org. Biomol. Chem., 18, 4046 - 4050 (2020), DOI:10.1039/D0OB00729C. ‡ These authors contributed equally.
  • R. A. Jagtap, S. K. Verma And B. Punji, MnBr2-Catalyzed Direct and Site-Selective Alkylation of Indoles and Benzo[h]quinoline, Org. Lett., 22, 4643 - 4647 (2020), DOI:10.1021/acs.orglett.0c01398.
  • R. A. Jagtap, P. P. Samal, C. P. Vinod, S. Krishnamurty And B. Punji, Iron-Catalyzed C(sp2)-H Alkylation of Indolines and Benzo[h]quinoline with Unactivated Alkyl Chlorides through Chelation-Assistance, ACS Catal., 10, 7312 - 7321 (2020), DOI:10.1021/acscatal.0c02030.
  • Paresh R. Athawale, Hanuman P. Kalmode, Zenia Motiwala, Kiran A. Kulkarni And D. Srinivasa Reddy, Overturning the Peribysin Family Natural Products Isolated from Periconia byssoides OUPS-N133: Synthesis and Stereochemical Revision of Peribysins A, B, C, F, and G, Organic Letters., 22, 3104 - 3109 (2020), DOI:10.1021/acs.orglett.0c00857.
  • Pronay Das, Gianluigi Lauro, Raffaele Riccio, D. Srinivasa Reddy And Giuseppe Bifulco, DFT/NMR Approach for the Configuration Assignment of Groups of Stereoisomers by the Combination and Comparison of Experimental and Predicted Sets of Data, Search Results Web result with site links The Journal of Organic Chemistry., 85, 3297 - 3306 (2020), DOI:10.1021/acs.joc.9b03129.
  • D. K. Pandey, A. B. Shabade And B. Punji, Copper-Catalyzed Direct Arylation of Indoles and Related (Hetero)arenes: A Ligandless and Solvent-free Approach, Adv. Synth. Catal., 362, 2534 - 2540 (2020).
  • B. Punji, B. Senthilkumar And C. V. Ramana, A Process for the Asymmetric Synthesis of SITAGLIPTIN Intermediate, Patent filed., , (2020).
  • D. M. Sharma And B. Punji, 3d Transition Metal Catalyzed Hydrogenation of Nitriles and Alkynes, Chem. Asian J., 15, 690 - 708 (2020), DOI:10.1002/asia.201901762.
  • R. A. Jagtap And B. Punji, C-H Functionalization of Indoles by 3d Transition-Metal Catalysis, Asian J. Org. Chem., 9, 326 - 342 (2020), DOI:10.1002/ajoc.201900554.
  • R. A. Jagtap And B. Punji, Nitrogen Ligands in Carbon-Carbon Bond Forming Reactions, Book Chapter., , (2020), DOI:John Wiley & Sons, Inc., of 111 River Street, Hoboken, NJ.
  • Cao, W.; Senthilkumar, B.; Causin, V.; Swamy, V. P.; Wang, Y.; Saielli And G, Influence of the ion size on the stability of the smectic phase of ionic liquid crystals, Soft Matter., 16, 411 - 420 (2020).
  • Amol B. Viveki, Dnyaneshwar N. Garad, Rajesh G. Gonnade And Santosh B. Mhaske, "para-Selective copper-catalyzed C(sp2)–H amidation/dimerization of anilides via a radical pathway", Chem. Commun., 56, 1565 (2020).
  • Kishor V. Khopade, Anirban Sen, Rajkumar S. Birajdar, Uday P. Paulbudhe, Dattatry S. Kavale, Prashant S. Shinde And Dr. Santosh B. Mhaske and Dr. Samir H. Chikkali, "Highly Enantioselective Synthesis of Sitagliptin", Asian J. Org.Chem., 9, 189 - 191 (2020).
  • Thanusha Thatikonda, Siddharth K. Deepake And Utpal Das*, alpha-Angelica Lactone in a New Role: Facile Access to N-Aryl Tetrahydroisoquinolinones and Isoindolinones via Organocatalytic alpha-CH2 Oxygenation, Organic Letters., 21, 2532 - 2535 (2019), DOI:10.1021/acs.orglett.9b00224.
  • Someshwar B. Kale, Popat K. Jori, Thanusha Thatikonda, Rajesh G. Gonnade And Utpal Das*, 1,6-Conjugate-Addition-Induced [2 + 1] Annulation of para-Quinone Methides and Pyrazolones: Synthesis of Bis-Spiro Compounds with Contiguous Quaternary Spiro-Centers, Organic Letters., 21, 7736 - 7740 (2019), DOI:10.1021/acs.orglett.9b02641.
  • A. A. Wagh And M. Fernandes, 2’-5’-Isomerically Linked Thrombin-Binding Aptamer (isoTBA) Forms a Stable Unimolecular Parallel G-Quadruplex in the Presence of Sr2+ Ions, ChemistrySelect., 4, 10668 - 10673 (2019).
  • A. K. Yadav, H. Chilukuri, L. R. Kumari, M. Karthikeyan And M. Fernandes, p-Nitrophenylcarbonates: A New Class of Compounds for Chemodosimetric Colorimetric Fluoride Anion Sensing Detectable by the Naked Eye, ChemistrySelect., 4, 1830 - 1833 (2019).
  • Hanuman P Kalmode, Suhag S Patil, Kishor L Handore, Paresh R Athawale, Rambabu Dandela, Abhishek K Verma And Anirban Basu and D Srinivasa Reddy, Neural Anti?inflammatory Natural Product Periconianone A: Total Synthesis and Biological Evaluation, Eur. J. Org. Chem., , 2376 - 2381 (2019).
  • Kishor L. Handore, Hanuman P. Kalmode, Shahebaz Sayyad, B. Seetharamsingh, Ganesh Gathalkar, Sarang Padole, Pushpa V. Pawar, Mary Joseph And Avalokiteswar Sen and D. Srinivasa Reddy, Insect-Repellent and Mosquitocidal Effects of Noreremophilane- and Nardoaristolone-Based Compounds, ACS Omega., 4, 2188 - 2195 (2019).
  • Das TK, Ghosh A, Balanna K, Behera P, Gonnade RG, Marelli UK, Das AK And Biju AT, N-Heterocyclic Carbene-Catalyzed Umpolung of Imines for the Enantioselective Synthesis of Dihydroquinoxalines, ACS Catal., 9, 4065 - 4071 (2019), DOI:https://doi.org/10.1021/acscatal.9b00737.
  • Reichart F, Maltsev OV, Kapp TG, Räder AFB, Weinmüller M, Marelli UK, Notni J, Wurzer A, Beck R, Wester HJ, Steiger K, Di Maro S, Di Leva FS, Marinelli L, Nieberler M, Reuning U, Schwaiger M And Kessler H, Selective Targeting of Integrin ?v?8 by a Highly Active Cyclic Peptide, J. Med. Chem., 62, 2024 - 2037 (2019), DOI:https://doi.org/10.1021/acs.jmedchem.8b01588.
  • Tharun K. Kotammagari And Sayantan Paul and Asish K. Bhattacharya, Unusual Epimerization in Styryllactones: Synthesis of (?)-5- Hydroxygoniothalamin, (?)-5-Acetylgoniothalamin, and O?TBSGoniopypyrone, ACS Omega., 4, 22549 - 22556 (2019), DOI:DOI: 10.1021/acsomega.9b03263.
  • Sachin B. Agawane, Vidya S. Gupta, Mahesh J. Kulkarni, Asish K. Bhattacharya And Santosh S. Koratkar, Chemo-biological evaluation of antidiabetic activity of Mentha arvensis L. and its role in inhibition of advanced glycation end products, Journal of Ayurveda and Integrative Medicine., 10, 166 - 170 (2019), DOI:http://dx.doi.org/10.1016/j.jaim.2017.07.003.
  • Sachin B. Agawane, Vidya S. Gupta, Mahesh J. Kulkarni, Asish K. Bhattacharya, Santosh S. Koratkar And Vamkudoth Koteswara Rao, Patho-physiological evaluation of Duranta erecta for the treatment of urolithiasis, Journal of Ayurveda and Integrative Medicine., 10, 4 - 11 (2019), DOI:http://dx.doi.org/10.1016/j.jaim.2017.08.001.
  • Eswar K Aratikatla And and Asish K. Bhattacharya, A Short Review on Synthetic Routes of Antiepileptic Drug (R)-Lacosamide, Org. Process Res. Dev., , 1 - 20 (2019), DOI:DOI: 10.1021/acs.oprd.9b00373.
  • Hemender R. Chand and Asish K. Bhattacharya, Hemiketal-Keto Tautomerism in 2-Deoxy-?-lactones Mediated by 2-Lithiothiazole in Solution State: A Formal Synthesis of DAH, Kamusol and Their C5 Epimers, Asian J. Org. Chem., 8, 2113 - 2120 (2019), DOI:DOI: 10.1002/ajoc.201900407.
  • Deepti Kalsi, Nagaraju Barsu, Sagnik Chakrabarti, Pardeep Dahiya, Magnus Rueping And and Basker Sundararaju, C–H and N–H bond annulation of aryl amides with unactivated olefins by merging cobalt (III) and photoredox catalysis, Chem. Commun., 55, 11626 - 11629 (2019), DOI:DOI https://doi.org/10.1039/C9CC05744G.
  • Pawan S. Dhote And Chepuri V. Ramana*, One-pot Au [III]-/Lewis acid catalyzed cycloisomerization of nitroalkynes and [3+ 3] cycloaddition with donor–acceptor cyclopropanes, Org. Lett., 21, 6221 - 6224 (2019), DOI:org/10.1021/acs.orglett.9b02035.
  • Kolluru Srinivas, Shaziya K. Siddiqui, Jyoti Mudaliar And Chepuri V. Ramana*, Ru (II)-catalyzed C–H activation/alkylation of 3-formylbenzofurans with conjugated olefins: product divergence, J. Org. Chem., 84, 5056 - 5066 (2019), DOI:10.1021/acs.joc.8b03267.
  • Abdul Motaleb, Soniya Rani, Tamal Das, Rajesh G Gonnade And Pradip Maity*, Phosphite Catalyzed C–H Allylation of Azaarenes via an Enantioselective [2,3]-Aza-Wittig Rearrangement, Angew. Chem. Int. Ed., 58, 14014 - 14109 (2019), DOI:10.1002/anie.201906681.
  • Samantha L. Maki, Pradip Maity, Shannon Dougherty, Jennifer Johns And Salvatore D. Lepore*, Allenoate Prenucleophiles: A Triply Diastereoselective Approach to ?-Hydroxy Esters Containing All-Carbon ?-Quaternary Centers, Org. Lett., 21, 7952 - 7955 (2019), DOI:10.1021/acs.orglett.9b02930.
  • Banerjee, S.; Senthilkumar, B.; Patil And N. T, Gold-Catalyzed 1,2-Oxyalkynylation of N-Allenamides with Ethylnylbenziodoxolones, Org. Lett., 21, 1, 180 - 184 (2019), DOI:10.1021/acs.orglett.8b03651.
  • Milind M. Ahire, Mahesh D. Pol Dattatry, S. Kavale, Rajesh G. Gonnade And Santosh B. Mhaske, "Stereoselective construction of deoxy-cruciferane alkaloids by NHC-catalyzed intramolecular annulation of homoenolate with quinazolinone", Org. Biomol. Chem., 17, 7135 - 7139 (2019).
  • Garad D. N.; Mhaske S. B.* , “Ru-Catalyzed Regioselective Cascade Annulation of Acrylamides with 2-Alkynoates for the Synthesis of Various 6-Oxo Nicotinic Acid Esters”, J. Org. Chem., 84, 1863 - 1870 (2019).
  • Halder P.; Humne T. V.; Mhaske S. B.* , “Transition-Metal-Free Regioselective One-Pot Synthesis of Aryl Sulfones from Sodium Sulfinates via Quinone Imine Ketal”, J. Org. Chem., 84, 1372 - 1378 (2019).
  • Gorakhnath R. Jachak, Paresh R. Athawale, Rahul Choudhury, K. Kashinath And D. Srinivasa Reddy, Access to a Stereoisomer Library of Solomonamide Macrocycles, Chem. Asian J., 2019, 4572 - 4576 (2019), DOI:10.1002/asia.201901075.
  • Ramana Sreenivasa Rao, Femil Joseph Shajan And D. Srinivasa Reddy, A route to access imidazol[1,5-a]indole-1,3-diones and pyrrolo[1,2-c]imidazole-1,3-diones†, Org. Biomol. Chem., 2019, 8384 - 8390 (2019), DOI:10.1039/c9ob01462d.
  • Paresh R. Athawale, Neeta Kumari, Monica R. Dandawate, K. Kashinath And D. Srinivasa Reddy, Synthesis of Chiral Tetrahydrofuran Building Blocks fromPantolactones: Application in the Synthesis of Empagliflozinand Amprenavir Analogs, Eur. J. Org. Chem., 2019, 4805 - 4810 (2019), DOI:10.1002/ejoc.201900718.
  • Kishor L. Handore, Hanuman P. Kalmode, Shahebaz Sayyad, B. Seetharamsingh, Ganesh Gathalkar, Sarang Padole, Pushpa V. Pawar, Mary Joseph, Avalokiteswar Sen And D. Srinivasa Reddy, Insect-Repellent and Mosquitocidal Effects of Noreremophilane- and Nardoaristolone-Based Compounds, ACS Omega., 4(1), 2188 - 2195 (2019), DOI:https://doi.org/10.1021/acsomega.8b03652.
  • Ganesh S. Ghotekar, Devidas A. More, Viswanadh Nalla And M. Muthukrishnan*, A new enantioselective synthesis of antiobesity drug lorcaserin, New Journal of Chemistry., 43, 16876 - 16880 (2019), DOI:10.1039/C9NJ04234B.
  • Devidas A. More, Ganesh H. Shinde, Aslam C. Shaikh And M. Muthukrishnan*, Oxone promoted dehydrogenative Povarov cyclization of N-aryl glycine derivatives: an approach towards quinoline fused lactones and lactams†, RSC Advances., 9, 30277 - 30291 (2019), DOI:10.1039/C9RA06212B.
  • Ganesh S. Ghotekar, M. Mujahid And M. Muthukrishnan*, Efficient Synthesis of Optically Active Neolignans Ligraminol D and E, Synthesis., 51, 4291 - 4295 (2019), DOI:10.1055/s-0037-1611919.
  • Ganesh S. Ghotekar, Aslam C. Shaikh And M. Muthukrishnan*, Transition-Metal-Free Benzannulation of Tricarbonyl Derivatives with Arynes: Access to 1,3-Dinaphthol Precursors for the Synthesis of Rhodamine Dye Analogues, The Journal of Organic Chemistry., 84, 2269 - 2276 (2019), DOI:10.1021/acs.joc.8b02560.
  • Ganesh S. Ghotekar, Mohammad Mujahid And M. Muthukrishnan*, Total Synthesis of Marine Natural Products Serinolamide A and Columbamide D, ACS Omega., 4, 1322 - 1328 (2019), DOI:10.1021/acsomega.8b03417.
  • D. K. Pandey, S. B. Ankade, A. Ali, C. P. Vinod And B. Punji, Nickel-Catalyzed C–H Alkylation of Indoles with Unactivated Alkyl Chlorides: Evidence of Ni(I)/Ni(III) Pathway, Chem. Sci., 10, 9493 - 9500 (2019).
  • U. N. Patel, R. A. Jagtap And B. Punji, Scope and Mechanistic Aspect of Nickel-Catalyzed Alkenylation of Benzothiazoles and Related Azoles with Styryl Bromides, Organometallics., 38, 2422 - 2430 (2019).
  • D. M. Sharma And B. Punji, Selective Synthesis of Secondary Amines from Nitriles by a User-Friendly Cobalt Catalyst, Adv. Synth. Catal., 361, 3930 - 3936 (2019).
  • D. K. Pandey, M. Vijaykumar And B. Punji, Nickel-Catalyzed C(2)-H Arylation of Indoles with Aryl Chlorides under Neat Condition, J. Org. Chem., 84, 12800 - 12808 (2019).
  • Yeware Amar, Agrawal Sonia And Sarkar Dhiman, A high content screening assay for identifying inhibitors against active and dormant state intracellular Mycobacterium tuberculosis, Journal of Microbiological Methods., 164, 105687 (2019).
  • Yeware Amar , Gample Suwarna, Agrawal Sonia And Sarkar Dhiman, Using diphenyleneiodonium to induce a viable but non-culturable phenotype in Mycobacterium tuberculosis and its metabolomics analysis, PLoS One., 14:8, e0220628 (2019).
  • Gample Suwarna, Agrawal Sonia And Sarkar Dhiman, Evidence of nitrite acting as a stable and robust inducer of non-cultivability in Mycobacterium tuberculosis with physiological relevance, Scientific reports., 9:1, 9261 (2019).
  • Uttam B Karale, Vagolu Siva Krishna, E Vamshi Krishna, Amit S Choudhari, Manjulika Shukla, Vikas R Gaikwad, B Mahizhaveni, Sidharth Chopra, Sunil Misra, Dhiman Sarkar, Dharmarajan Sriram, VN Azger Dusthackeer And Haridas B Rode, Synthesis and biological evaluation of 2, 4, 5-trisubstituted thiazoles as antituberculosis agents effective against drug-resistant tuberculosis, European journal of medicinal chemistry., , (2019).
  • Vikas Shinde, Pramod Mahulikar, Pravin C Mhaske, Shakti Chakraborty, Amit Choudhari, Siddharth Phalle, Prafulla Choudhari And Dhiman Sarkar, Synthesis and antimycobacterial evaluation of new 5-(1-benzyl-1H-1,2,3-triazol-4-yl)-4-methyl-2-arylthiazole derivatives, Medicinal Chemistry Research., 28, 805 - 819 (2019).
  • Sushma J Takate, Abhijit D Shinde, Bhausaheb K Karale, Hemant Akolkar, Laxman Nawale, Dhiman Sarkar And Pravin C Mhaske, Thiazolyl-pyrazole derivatives as potential antimycobacterial agents, Bioorganic & medicinal chemistry letters., 29, 1199 - 1202 (2019).
  • Atmaram Upare A, Gadekar PK, Sivaramakrishnan H, Naik N3, Khedkar VM, Sarkar D, Choudhari A And Mohana Roopan S, Design and Synthesis of 2?Amino?thiophene?proline?conjugates and Their Anti?tubercular Activity against Mycobacterium Tuberculosis H37Ra, Bioorg Chem., 86, 507 - 512 (2019), DOI:doi: 10.1016/j.bioorg.2019.01.054.
  • Vidya B. Gunjal And D. Srinivasa Reddy, Total synthesis of Met10-teixobactin, Tetrahedron Letters., 60, 1909 - 1912 (2019), DOI:doi.org/10.1016/j.tetlet.2019.06.027.
 
 


News, Events and Highlights

Recent Publications        view all>>

Announcements