Research Group Publications

  • Vinita Yadav, Ekambaram Balaraman And Santosh B. Mhaske, Phosphine-Free Manganese(II)-Catalyst Enables Acceptorless Dehydrogenative Coupling of Alcohols with Indoles, Advanced Synthesis & Catalysis., 363, (2021), DOI:
  • Amol B. Viveki, § Mahesh D. Pol, § Priyanka Halder, Sameer R. Sonavane And Santosh B. Mhaske*, Annulation of Enals with Carbamoylpropiolates via NHC-Catalyzed Enolate Pathway: Access to Functionalized Maleimides/Iso-maleimides and Synthesis of Aspergillus FH-X-213, J. Org. Chem., 86,14, 9466 - 9477 (2021), DOI:
  • Rajeshwari Tiwari, Prashant Suresh Shinde, Sreejesh Sreedharan, Anik Kumar Dey, Katherine Vallis, Santosh B. Mhaske, Sumit Kumar Pramanik And Amitava Das, "Photoactivable Prodrug for Simultaneous Release of Mertansine, and CO along with a BODIPY Derivative as a Luminescent Marker in Mitochondria: A Proof of Concept for NIR Image-Guided Cancer Therapy", Chemical Science., Just Accepted, (2020).
  • Priyanka Halder, Mahesh D. Pol, Milind M Ahire And Santosh B. Mhaske , "Construction of Unique SCF3-Containing Building Blocks via Allylic Alkylation of Morita-Baylis-Hillman Adducts", Org. Biomol. Chem., 18, 2085 - 2093 (2020).
  • Amol B. Viveki, Dnyaneshwar N. Garad, Rajesh G. Gonnade And Santosh B. Mhaske, "para-Selective copper-catalyzed C(sp2)–H amidation/dimerization of anilides via a radical pathway", Chem. Commun., 56, 1565 (2020).
  • Kishor V. Khopade, Anirban Sen, Rajkumar S. Birajdar, Uday P. Paulbudhe, Dattatry S. Kavale, Prashant S. Shinde And Dr. Santosh B. Mhaske and Dr. Samir H. Chikkali, "Highly Enantioselective Synthesis of Sitagliptin", Asian J. Org.Chem., 9, 189 - 191 (2020).
  • Milind M. Ahire, Mahesh D. Pol Dattatry, S. Kavale, Rajesh G. Gonnade And Santosh B. Mhaske, "Stereoselective construction of deoxy-cruciferane alkaloids by NHC-catalyzed intramolecular annulation of homoenolate with quinazolinone", Org. Biomol. Chem., 17, 7135 - 7139 (2019).
  • Garad D. N.; Mhaske S. B.* , “Ru-Catalyzed Regioselective Cascade Annulation of Acrylamides with 2-Alkynoates for the Synthesis of Various 6-Oxo Nicotinic Acid Esters”, J. Org. Chem., 84, 1863 - 1870 (2019).
  • Halder P.; Humne T. V.; Mhaske S. B.* , “Transition-Metal-Free Regioselective One-Pot Synthesis of Aryl Sulfones from Sodium Sulfinates via Quinone Imine Ketal”, J. Org. Chem., 84, 1372 - 1378 (2019).
  • Ahire M. M.; Mhaske S. B.* , “Isa-NHC-catalyzed intermolecular Stetter reaction of aromaticaldehydes with maleimides: An efficient access to 3-aroylsuccinimides”, Tetrahedron., 74, 2079 - 2084 (2018).
  • Mahajan P. S.; Mhaske S. B.* , “Silver-Mediated Oxidative Decarboxylative Intramolecular Asymmetric Radical Cyclization (Csp3–Csp2) via Memory of Chirality: Access to Circumdatin Alkaloids”, Org. Lett., 20, 2092 - 2095 (2018).
  • Viveki A. B.; Mhaske S. B* , “Ruthenium-Catalyzed Regioselective Alkenylation/Tandem Hydroamidative Cyclization of Unmasked Quinazolinones Using Terminal Alkynes”, J. Org. Chem., 83, 8906 - 8913 (2018).
  • Pandya V. G.; Mhaske S. B*, “Divergent Synthesis of Oxindolylidene Acetates and Spirooxindolopyrrolidones from Arynes”, Org. Lett., 20, 1483 - 1486 (2018).
  • Ahire M. M.; Thoke M. B.; Mhaske S. B* , “Application of Sulfur Ylides in 1,2-Difunctionalization of Arynes via Insertion into C–S ?-Bond”, Org. Lett., 20, 848 - 851 (2018).
  • Dhokale R. A.; Mhaske S. B*, “Transition-Metal-Catalyzed Reactions Involving Arynes”, Synthesis., 50, 1 - 16 (2018).
  • Ahire M. M.; Mhaske S. B*, “Synthesis of Succinimide Derivatives by NHC-Catalyzed Stetter Reaction of Aromatic Aldehydes with N-Substituted Itaconimides”, ACS Omega., 2, 6598 - 6604 (2017).
  • Garad D. N.; Viveki A. B.; Mhaske S. B*, “Pd-Catalyzed Regioselective Mono-Arylation: Quinazolinone as the Inherent Directing Group for C(sp2)–H Activation”, J. Org. Chem., 82, 6366 - 6372 (2017).
  • Garad D. N.; Mhaske S. B*, “Diversification of Quinazolinones by Pd-Catalyzed C(sp3)-Acetoxylation”, J. Org. Chem., 82, 10470 - 10478 (2017).
  • Dhokale R. A.; Mhaske S. B*, “Diversity-oriented Synthesis of Spiroannulated Benofuran-3-one Scaffold of Leptosphaerin C and Congeners via Aryne insertion”, J. Org. Chem., 82, 4875 - 4882 (2017).
  • Mahajan J. P.; Mhaske S. B*. , “Synthesis of Methyl-Protected (±)-Chlorizidine A”, Org. Lett., 19, 2774 - 2776 (2017).
  • Divse J. M.; Mhaske S. B.; Charolkar C. R.; Sant D. G.; Tupe S. G.; Deshpande M. V.; Khedkar V. M.; Nawale L. U.; Sarkar D.; Pore V. S.*, “Synthesis and biological evaluation of new fluconazole b-lactam conjugates linked via 1,2,3-triazole”, New J. Chem., 41, 470 - 479 (2017).
  • Ahire M. M.; Khan R.; Mhaske S. B*, “Synthesis of o-Methyl Trifluoromethyl Sulfide Substituted Benzophenones via 1,2-Difunctionalization of Aryne by Insertion into the C–C Bond”, Org. Lett., 19, 2134 - 2137 (2017).
  • Mahajan P. S.; Humne V. T.; Mhaske S. B*, “Achmatowicz Reaction: A Versatile Tool in Bioactive Natural Products Synthesis”, Curr. Org. Chem., 21, 503 - 545 (2017).
  • Garad D. N.; Mhaske S.B.* , “Pd(II)-Catalyzed Intramolecular Tandem Olefin Amidation/C–H Activation Protocol for the Syntheses of the Protoberberine Class of Natural Products”, Org. Lett., 18, 3862 - 3865 (2016).
  • Agarwalla H.; Mahajan P. S.; Sahu D.; Taye N.; Ganguly B.; Mhaske S. B.*; Chattopadhyay S.; Das A.*, “A Switch-On NIR Probe for Specific Detection of Hg2+ Ion in Aqueous Medium and in Mitochondria”, Inorg. Chem., 55, 12052 - 12060 (2016).
  • Dhokale R. A. and Mhaske S. B*, “Nucleophilic Nitration of Arynes by Sodium Nitrite and its Multicomponent Reaction Leading to Double-Functionalized Arenes”, Org.Lett., 18, 3010 (2016).
    (Most read article in July 2016)
  • Mahajan, P. S.; Humne, V. T.; Tanpure And S. D. and Mhaske S. B*, “Radical Beckmann Rearrangement and Its Application in the Formal Total Synthesis of Antimalarial Natural Product Isocryptolepine via C-H Activation”, Org. Lett., 18, 3450 - 3453 (2016).
  • Franke J.; Bock M.; Dehn R.; Fohrer J.; Mhaske S. B.; Migliorini A.; Kanakis A. A.; Jansen R.; Herrmann J.; Müller R.; Kirschning A., Total and Semi?Syntheses of Antimicrobial Thuggacin Derivatives, Chem. Eur. J., 21, 4272 - 4284 (2015).
  • Garad D. N.; Tanpure S. D. and Mhaske S.B. , “Radical-mediated dehydrative preparation of cyclic imides using (NH4)2S2O8–DMSO: application to the synthesis of vernakalant”, J. Org. Chem., 11, 1008 - 1016 (2015).
  • Mahajan, P. S.; Tanpure, S. D.; More, N. A.; Gajbhiye And J. M. and Mhaske S. B*, “Ammonium persulfate activated DMSO as a one-carbon synthon for the synthesis of methylenebisamides and other applications”, RSC Adv., 5, 101641 - 101646 (2015).
  • Pandya V. G. and Mhaske S. B*, “Transition-Metal-Free C–S Bond Formation: A Facile Access to Aryl Sulfones from Sodium Sulfinates via Arynes”, Org. Lett., 16, 3836 (2014).
    (Highlighted in Organic Portal) (Most read article in July 2014)
  • Mahajan P. S.; Gonnade R. G. and Mhaske S. B*., “Protecting-Group-Free Diastereoselective Total Synthesis of (±)-6-epi-Cleistenolide and Chemoenzymic Synthesis of (–)-6-epi-Cleistenolide”, Eur. J. Org. Chem., , 8049 - 8054 (2014).
  • Mahajan P. S.; Mahajan J. P. and Mhaske S. B* , Malonic ester amide synthesis. An efficient methodology for synthesis of amides, Synth. Commun., 43, 2508 - 2516 (2013).
  • P. S. Mahajan, J. P. Mahajan And S. B. Mhaske, Malonic Ester Amide Synthesis: An Efficient Amide Synthesis Methodology, Synth. Commun., , (2012).
  • J. P. Mahajan, Y. R. Suryawanshi And S. B. Mhaske, Pd-Catalyzed C-H Activation: Synthesis of Antimalarial Natural Products Marinoquinoline A, Aplidiopsamine A and their Potential Hybrid NCLite-M1, Org. Lett., , (2012).
    Manuscript ready for communication to Org. Lett.
  • R. A. Dhokale, P. R. Thakare And S. B. Mhaske, Transition-Metal-Free C-Arylation at Room Temperature by arynes, Org. Lett., 14, 3994 (2012).
  • Dhokale R. A. And Mhaske S. B* , P-Arylation: Arynes to Aryl Phosphonates, -Phosphinates, Phosphine oxides, Org.Lett., 15, 2218 (2012).
    (Highlighted in Organic Chemistry Portal)
  • S. B. Mhaske, Using continuous flow process in the chemical industry, Chemical Industry Digest., ?24, 89 (2011).
    ? Invited article
  • U. A. Kshirsagar, S. B. Mhaske And N. P. Argade, Hexamethyldisilazane-iodine induced intramolecular dehydrative cyclization of diamides: a general access to natural and unnatural quinazolinones, Tetrahedron Lett., 48, 3243 (2007).
  • H.-S. Chong, S. B. Mhaske, M. Lin, S. Bhuniya, H. A. Song, M. W. Brechbiel And X. Sun, Novel synthetic ligands for targeted PET imaging and radiotherapy of copper, Bioorg. & Med. Chem. Lett., 17, 6107 (2007).
  • ? S. B. Mhaske And N. P. Argade, The chemistry of recently isolated naturally occurring quinazolinone alkaloids, Tetrahedron., 62, 9787 (2006).
    Recognized as ?Top-25 most downloaded article? 2006
  • K. P. Haval, S. B. Mhaske And N. P. , Cyanuric chloride: Decent dehydrating agent for an exclusive and efficient synthesis of kinetically controlled isomaleimides, Tetrahedron., 62, 937 (2006).
  • S. B. Mhaske, Mesityllithium, Synlett ., 184, (2005).
    (spotlight 108)
  • S. B. Mhaske And N. P. Argade, Regioselective quinazolinone-directed ortho lithiation of quinazolinoylquinoline: Practical synthesis of naturally occurring human DNA topoisomerase I poison luotonin A and luotonins B and E, J. Org. Chem., 69, 4563 (2004).
    ?Dr. Rajappa Award? for ?Best Research Paper?
  • S. B. Mhaske. N. P. Argade, Facile zeolite induced Fischer-indole synthesis: A new approach to bioactive natural product rutaecarpine, Tetrahedron ., 60, 3417 (2004).
  • M. K. Sahoo, S. B. Mhaske And N. P. Argade, Facile routes to alkoxymaleimides/maleic anhydrides, Synthesis., 346, (2003).
  • S. B. Mhaske And N. P. Argade, Base-induced alcoholysis of N-arylmaleimides: Facile in situ oxa-Michael addition to alkyl maleanilates: Two-step one-pot rapid access to alkoxysuccinic acids, Synthesis., 863, (2003).
  • F. S. B. Mhaske And N. P. Argade, Biogenetic synthesis of luotonin, Synthesis., 323, (2002).
  • S. B. Mhaske And N. P. Argade, Concise and efficient synthesis of bioactive natural products pegamine, deoxyvasicinone and (-)-vasicinone, J. Org. Chem., 66, 9038 (2001).
  • S. B. Mhaske, R. V. Bhingarkar, M. B. Sabne, R. Mercier And S. P. Vernekar , Synthesis and characterization of end-capped polyimides and their Gas permeability properties, J. Appl. Polym. Sci., 77, 627 (2000).
  • X. Ma, H. A. Song, H. Lee, S. B. Mhaske, S. Bhuniya And H.-S. Chong, Generation of new chelates for targeted MRI and radioimmuniotherapy, , (0000).
    . Abstracts of Papers, 233rd ACS National Meeting, Chicago, IL, United States, March 25-29, 2007, Abstract No. MEDI-101.
  • ? H.-S. Chong; H. A. Song; X. Ma; S. Lim; X. Sun; S. B. Mhaske, Bile acid-based polyaminocarboxylate conjugates as targeted antitumor agents, , (0000).
    Abstracts of Papers, 238th ACS National Meeting, Washington, DC, United States, August 16-20, 2009, Abstract No. MEDI-310.